SCHEMBL24136167

SCHEMBL24136167

COc1ccc(F)c2c1cc(C#N)n2I

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.37
IMPDH1 P20839 1/20 0.37
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
NAAA Q02083 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NQO1 P15559 1/20 0.32
S1PR3 Q99500 3/20 0.31
AR P10275 3/20 0.31
S1PR1 P21453 1/20 0.31
EGFR P00533 2/20 0.31
ERBB2 P04626 2/20 0.31
SRC P12931 1/20 0.31
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22434808 0.84 IMPDH2 (0.38) IMPDH2IMPDH1KDM4EUSP2ALDH1A1
SCHEMBL24136189 0.78 MEN1 (0.35) KDM4EALDH1A1MEN1KMT2ANQO1
SCHEMBL24136204 0.77 L3MBTL1 (0.35) ALDH1A1MEN1KMT2ANQO1LMNA
SCHEMBL24136211 0.73 IMPDH2 (0.39) IMPDH2IMPDH1KDM4EALDH1A1MEN1
SCHEMBL20505499 0.71 KMT2A (0.34) KMT2ALMNAMAPK1HTTRAB9A
SCHEMBL28479024 0.71 KMT2A (0.32) KDM4EALDH1A1KMT2ALMNAMAPK1
SCHEMBL24136165 0.71 SLC6A3 (0.32) IMPDH2IMPDH1KDM4EUSP2ALDH1A1
SCHEMBL22434645 0.69 PGR (0.34) AR
SCHEMBL22434669 0.67 CYP19A1 (0.40) KDM4EALDH1A1MEN1KMT2ANQO1
SCHEMBL24136181 0.67 AR (0.30) KDM4EALDH1A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3928836-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS Idorsia Pharmaceuticals Ltd (CH) 2021-12-29 EP disclosed