SCHEMBL6286018

SCHEMBL6286018

CC(C)(C)OC(=O)Nc1ccc[nH]c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
RXFP1 Q9HBX9 1/20 0.44
KDM4E B2RXH2 3/20 0.42
GAA P10253 3/20 0.42
BLM P54132 3/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 2/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
THRB P10828 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 1/20 0.42
METAP1 P53582 1/20 0.41
ALPL P05186 1/20 0.41
CDC25A P30304 1/20 0.41
CDC25B P30305 1/20 0.41
TSHR P16473 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2880191 0.79 LMNA (0.54) RAB9ANPC1SMN1; SMN2RXFP1GAA
SCHEMBL17390354 0.79 RXFP1 (0.40) RAB9ANPC1SMN1; SMN2RXFP1KDM4E
SCHEMBL5777669 0.79 JAK1 (0.39) RAB9ANPC1SMN1; SMN2RXFP1GAA
SCHEMBL1566862 0.79 RAB9A (0.52) RAB9ANPC1SMN1; SMN2RXFP1GAA
SCHEMBL21481533 0.78 NR3C1 (0.52) RAB9ANPC1SMN1; SMN2RXFP1POLB
SCHEMBL24251779 0.78 BLM (0.42) KDM4EGAABLMKMT2APOLB
SCHEMBL6826283 0.76 ALDH1A1 (0.50) RAB9ANPC1KDM4EGAABLM
SCHEMBL718382 0.76 SIGMAR1 (0.49) RAB9ANPC1SMN1; SMN2RXFP1GAA
SCHEMBL7223042 0.75 CA12 (0.39) RXFP1GAAPOLBLMNAMETAP1
SCHEMBL23134022 0.75 RAB9A (0.46) RAB9ANPC1SMN1; SMN2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137677-A1 PROTACS USEFUL AGAINST THE MAIN PROTEASE SARS-COV-2 TOCRIS COOKSON LTD (GB) 2026-05-21 US disclosed
EP-4701735-A1 HETEROCYCLIC DERIVATIVE AS MITOGEN-ACTIVATED PROTEIN KINASE (MEK) INHIBITOR Nested Therapeutics, Inc. (US) 2026-03-04 EP disclosed
WO-2025226862-A1 CYCLIN INHIBITORS CIRCLE PHARMA, INC. (US) 2025-10-30 WO disclosed
US-20250289811-A1 HETEROCYCLIC DERIVATIVES AS MITOGEN-ACTIVATED PROTEIN KINASE (MEK) INHIBITORS NESTED THERAPEUTICS, INC. 2025-09-18 US disclosed
EP-4598914-A1 PROTACS USEFUL AGAINST THE MAIN PROTEASE SARS-COV-2 Tocris Cookson Limited (GB) 2025-08-13 EP disclosed
US-20250195495-A1 RNA Virus Inhibitor Compounds and Uses Thereof THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2025-06-19 US disclosed
CN-119954831-A Pyrimidopyrazoles, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2025-05-09 CN disclosed
EP-4514471-A1 HETEROCYCLIC DERIVATIVES AS MITOGEN-ACTIVATED PROTEIN KINASE (MEK) INHIBITORS Nested Therapeutics, Inc. (US) 2025-03-05 EP disclosed
US-12186309-B2 RNA virus inhibitor compounds and uses thereof THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2025-01-07 US disclosed
WO-2024226579-A9 HETEROCYCLIC DERIVATIVE AS MITOGEN-ACTIVATED PROTEIN KINASE (MEK) INHIBITOR NESTED THERAPEUTICS, INC. (US) 2024-12-26 WO disclosed
US-10562906-B2 TYK2 inhibitors and uses thereof Nimbus Lakshimi, Inc. (US) 2020-02-18 US disclosed
US-20190241576-A1 TYK2 INHIBITORS AND USES THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-08-08 US disclosed
WO-2019023468-A1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI, INC. (US) 2019-01-31 WO disclosed
US-20050165062-A1 Substituted polycyclic aryl and heteroaryl pyridones useful for selective inhibition of the coagulation cascade PHARMACIA CORPORATION (US) 2005-07-28 US disclosed
US-6870056-B1 Substitituted polycyclic aryl and heteroaryl pyridones useful for selective inhibition of the coagulation cascade PHARMACIA CORPORATION (US) 2005-03-22 US disclosed
US-6867217-B1 Substituted polycyclic aryl and heteroaryl pyridones useful for selective inhibition of the coagulation cascade PHARMACIA CORPORATION (US) 2005-03-15 US disclosed
CN-1378534-A Substituted polycyclic aryl and heteroaryl pyridones for selective inhibition of the coagulation cascade PHARMACIA CO (US) 2002-11-06 CN disclosed
EP-1178964-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL PYRIDONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE Pharmacia Corporation (US) 2002-02-13 EP disclosed
WO-2001087842-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL PYRIDONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2001-11-22 WO disclosed
WO-2000069826-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL PYRIDONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2000-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165062-A1 Substituted polycyclic aryl and heteroaryl pyridones useful for selective inhibition of the coagulation cascade TFPI, PLAT, TFPI2 RAB9A 4090/4885NPC1 3928/4885SMN1; SMN2 3799/4885
US-10562906-B2 TYK2 inhibitors and uses thereof TYK2, JAK2, JAK1 RAB9A 3462/4885NPC1 4595/4885SMN1; SMN2 1145/4885
US-20190241576-A1 TYK2 INHIBITORS AND USES THEREOF TYK2, JAK2, JAK1 RAB9A 3462/4885NPC1 4595/4885SMN1; SMN2 1145/4885
US-20250195495-A1 RNA Virus Inhibitor Compounds and Uses Thereof NSUN3, EIF2AK2, NSUN2 RAB9A 1943/4885NPC1 503/4885SMN1; SMN2 1395/4885
US-12186309-B2 RNA virus inhibitor compounds and uses thereof NSUN3, EIF2AK2, NSUN2 RAB9A 1943/4885NPC1 503/4885SMN1; SMN2 1395/4885
US-20260137677-A1 PROTACS USEFUL AGAINST THE MAIN PROTEASE SARS-COV-2 XIAP, MDM2, SARS1 RAB9A 1660/4885NPC1 3028/4885SMN1; SMN2 1397/4885
US-20250289811-A1 HETEROCYCLIC DERIVATIVES AS MITOGEN-ACTIVATED PROTEIN KINASE (MEK) INHIBITORS MAPK1, MAP3K1, MAPK3 RAB9A 914/4885NPC1 4497/4885SMN1; SMN2 4521/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.