SCHEMBL24327879

SCHEMBL24327879

CNc1nnc2c(-c3cnn(C)c3)nc(-c3ccc(C(F)(F)F)cc3)cn12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TEK Q02763 2/20 0.45
EPHB4 P54760 1/20 0.45
NPBWR1 P48145 1/20 0.39
SCD O00767 2/20 0.38
ADORA2A P29274 1/20 0.36
KDR P35968 2/20 0.36
TYK2 P29597 2/20 0.35
MET P08581 3/20 0.35
TLR8 Q9NR97 1/20 0.35
CHEK1 O14757 1/20 0.34
KCNH2 Q12809 1/20 0.34
PDE2A O00408 1/20 0.34
LRRK2 Q5S007 1/20 0.34
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
JAK3 P52333 1/20 0.33
BRD4 O60885 1/20 0.33
NQO2 P16083 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24327329 0.87 EPHB4 (0.42) TEKEPHB4NPBWR1SCDTYK2
SCHEMBL24327327 0.86 TEK (0.47) TEKEPHB4NPBWR1SCDADORA2A
SCHEMBL24327878 0.85 EPHB4 (0.42) TEKEPHB4NPBWR1SCDTYK2
SCHEMBL24328762 0.82 TRPV3 (0.40) TEKEPHB4SCDTYK2KCNH2
SCHEMBL24328759 0.76 TEK (0.41) TEKEPHB4NPBWR1SCDKDR
SCHEMBL24328751 0.75 IRAK1 (0.43) TEKEPHB4KDRTYK2CHEK1
SCHEMBL24328760 0.75 IRAK1 (0.43) TEKEPHB4KDRTYK2CHEK1
SCHEMBL24328734 0.75 IRAK1 (0.43) TEKEPHB4KDRTYK2CHEK1
SCHEMBL24327773 0.71 KCNH2 (0.55) TEKEPHB4NPBWR1KCNH2MAPK1
SCHEMBL24328691 0.71 EPHB4 (0.46) TEKEPHB4NPBWR1TYK2TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed