SCHEMBL24328743

SCHEMBL24328743

CN1C(=O)C(=C2CC(c3ccccc3)NN2)C(=O)N(C)C1=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.42
KMT2A Q03164 3/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HSD17B2 P37059 2/20 0.33
ALDH1A1 P00352 2/20 0.33
ATM Q13315 1/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24329754 0.93 BRD4 (0.42) BRD4KMT2ATSHRKDM4EHSD17B2
SCHEMBL24329187 0.89 KCNH2 (0.38) BRD4KMT2ALMNAMAPTALDH1A1
SCHEMBL29564321 0.87 TP53 (0.34) BRD4KMT2AMEN1LMNAMAPT
SCHEMBL29565262 0.86 ALDH1A1 (0.36) BRD4KMT2ATSHRSMN1; SMN2MEN1
SCHEMBL29564756 0.86 TDP1 (0.32) KMT2ATSHRMEN1LMNAHSD17B2
SCHEMBL24328744 0.84 MEN1 (0.39) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL24329099 0.84 KMT2A (0.40) KMT2ASMN1; SMN2MEN1LMNAMAPT
SCHEMBL24329665 0.79 BRD4 (0.40) BRD4KMT2ATSHRSMN1; SMN2MAPT
SCHEMBL24329755 0.78
SCHEMBL24328749 0.78 NPSR1 (0.46) LMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022080346-A1 NOVEL NITROGEN-CONTAINING CYCLIC COMPOUND AND APPLICATION THEREOF 国立大学法人佐賀大学 2022-04-21 WO disclosed