SCHEMBL24328744

SCHEMBL24328744

CN1C(=O)C(=C2CC(c3ccc4ccccc4c3)NN2)C(=O)N(C)C1=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
SLC6A4 P31645 4/20 0.36
SLC6A2 P23975 3/20 0.36
SLC6A3 Q01959 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
DRD2 P14416 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ACHE P22303 1/20 0.34
KCNH2 Q12809 1/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
ERBB3 P21860 1/20 0.33
KDR P35968 1/20 0.33
PTK2 Q05397 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24328743 0.84 BRD4 (0.42) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL24329754 0.84 BRD4 (0.42) KMT2AKDM4E
SCHEMBL24329187 0.82 KCNH2 (0.38) KMT2AALDH1A1HPGDKCNH2
SCHEMBL29564321 0.81 TP53 (0.34) MEN1KMT2AALDH1A1KDM4E
SCHEMBL24329099 0.80 KMT2A (0.40) MEN1KMT2AALDH1A1KDM4E
SCHEMBL29565262 0.80 ALDH1A1 (0.36) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL29564756 0.80 TDP1 (0.32) MEN1KMT2A
SCHEMBL24329733 0.74 ACHE (0.44) MEN1KMT2ASLC6A4SLC6A3ACHE
SCHEMBL24329755 0.72
SCHEMBL24329174 0.68 HTR2A (0.34) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022080346-A1 NOVEL NITROGEN-CONTAINING CYCLIC COMPOUND AND APPLICATION THEREOF 国立大学法人佐賀大学 2022-04-21 WO disclosed