SCHEMBL29565262

SCHEMBL29565262

CN1C(=O)C(=C2CC(c3ccc(Cl)cc3)NN2)C(=O)N(C)C1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
GAA P10253 1/20 0.36
CXCR5 P32302 1/20 0.36
APLNR P35414 1/20 0.36
CCR6 P51684 1/20 0.36
PTGS2 P35354 1/20 0.34
SRD5A1 P18405 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
LMNA P02545 4/20 0.33
THRB P10828 2/20 0.33
APEX1 P27695 2/20 0.33
PMP22 Q01453 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29564321 0.88 TP53 (0.34) ALDH1A1KDM4EMAPTGAAPTGS2
SCHEMBL29564756 0.86 TDP1 (0.32) TDP1GAALMNATSHRKMT2A
SCHEMBL24328743 0.86 BRD4 (0.42) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL24329754 0.85 BRD4 (0.42) KDM4EPTGS2TSHRKMT2ABRD4
SCHEMBL24329099 0.84 KMT2A (0.40) ALDH1A1KDM4ESMN1; SMN2MAPTGAA
SCHEMBL24329187 0.81 KCNH2 (0.38) ALDH1A1MAPTTDP1LMNATHRB
SCHEMBL24328744 0.80 MEN1 (0.39) ALDH1A1KDM4EKMT2AMEN1HPGD
SCHEMBL24329755 0.78
SCHEMBL24329174 0.73 HTR2A (0.34) ALDH1A1MAPTGAATSHR
SCHEMBL24328739 0.71 MAOA (0.40) ALDH1A1KDM4ESMN1; SMN2PTGS2GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022080346-A1 NOVEL NITROGEN-CONTAINING CYCLIC COMPOUND AND APPLICATION THEREOF 国立大学法人佐賀大学 2022-04-21 WO disclosed