SCHEMBL24329099

SCHEMBL24329099

COc1ccc(C2CC(=C3C(=O)N(C)C(=O)N(C)C3=O)NN2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
THRB P10828 1/20 0.39
PTGS2 P35354 2/20 0.39
PTGS1 P23219 1/20 0.39
MAPT P10636 3/20 0.38
LMNA P02545 1/20 0.38
ALDH1A1 P00352 4/20 0.36
GAA P10253 4/20 0.36
KDM4E B2RXH2 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
GLA P06280 1/20 0.36
MAP2K1 Q02750 1/20 0.35
HIF1A Q16665 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TP53 P04637 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
NR1H2 P55055 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24329187 0.86 KCNH2 (0.38) KMT2ATHRBMAPTLMNAALDH1A1
SCHEMBL29564321 0.85 TP53 (0.34) KMT2APTGS2MAPTLMNAALDH1A1
SCHEMBL29565262 0.84 ALDH1A1 (0.36) KMT2ATHRBPTGS2MAPTLMNA
SCHEMBL29564756 0.84 TDP1 (0.32) KMT2ALMNAGAAMEN1
SCHEMBL24328743 0.84 BRD4 (0.42) KMT2AMAPTLMNAALDH1A1KDM4E
SCHEMBL24329754 0.83 BRD4 (0.42) KMT2APTGS2KDM4ENR1H2NR1H3
SCHEMBL24328744 0.80 MEN1 (0.39) KMT2AALDH1A1KDM4EMEN1
SCHEMBL24329755 0.76
SCHEMBL24329174 0.74 HTR2A (0.34) MAPTALDH1A1GAA
SCHEMBL29564300 0.72 MAOA (0.42) KMT2APTGS2MAPTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022080346-A1 NOVEL NITROGEN-CONTAINING CYCLIC COMPOUND AND APPLICATION THEREOF 国立大学法人佐賀大学 2022-04-21 WO disclosed
WO-2022080346-A1 NOVEL NITROGEN-CONTAINING CYCLIC COMPOUND AND APPLICATION THEREOF 国立大学法人佐賀大学 2022-04-21 WO disclosed