SCHEMBL24329754

SCHEMBL24329754

CN1C(=O)C(=C2CC(c3ccc(-c4ccccc4)cc3)NN2)C(=O)N(C)C1=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.42
HSD17B2 P37059 3/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
PTGS2 P35354 1/20 0.34
PAX8 Q06710 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRNA7 P36544 1/20 0.32
BACE1 P56817 1/20 0.32
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
GSK3B P49841 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24328743 0.93 BRD4 (0.42) BRD4HSD17B2TSHRKMT2AKDM4E
SCHEMBL24329187 0.88 KCNH2 (0.38) BRD4KMT2ACHRNA7
SCHEMBL29564321 0.86 TP53 (0.34) BRD4PTGS2KMT2AKDM4E
SCHEMBL29564756 0.85 TDP1 (0.32) HSD17B2TSHRKMT2ABACE1MAOB
SCHEMBL29565262 0.85 ALDH1A1 (0.36) BRD4HSD17B2PTGS2TSHRKMT2A
SCHEMBL24328744 0.84 MEN1 (0.39) KMT2AKDM4E
SCHEMBL24329099 0.83 KMT2A (0.40) NR1H2NR1H3PTGS2KMT2AKDM4E
SCHEMBL24329755 0.80
SCHEMBL24329665 0.73 BRD4 (0.40) BRD4HSD17B2TSHRKMT2AKDM4E
SCHEMBL24328749 0.72 NPSR1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022080346-A1 NOVEL NITROGEN-CONTAINING CYCLIC COMPOUND AND APPLICATION THEREOF 国立大学法人佐賀大学 2022-04-21 WO disclosed
WO-2022080346-A1 NOVEL NITROGEN-CONTAINING CYCLIC COMPOUND AND APPLICATION THEREOF 国立大学法人佐賀大学 2022-04-21 WO disclosed