SCHEMBL24568636

SCHEMBL24568636

C=Cc1nc(-c2cc3ccc(OCc4ccccc4)nc3n2CC2CC2)c(C)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.34
ADORA1 P30542 3/20 0.34
SRC P12931 2/20 0.32
HCK P08631 1/20 0.32
CCNT1 O60563 1/20 0.32
CDK9 P50750 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32
CYP2D6 P10635 1/20 0.32
HRH1 P35367 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
ADORA2A P29274 2/20 0.32
APOBEC3G Q9HC16 1/20 0.31
PADI4 Q9UM07 1/20 0.31
MERTK Q12866 1/20 0.31
PDE5A O76074 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24568535 0.82 PADI4 (0.31) PADI4
SCHEMBL24568534 0.80 GRIA2 (0.32) PADI4
SCHEMBL24568632 0.78 NR1H2 (0.35)
SCHEMBL24568637 0.78 PADI4 (0.30) PADI4
SCHEMBL24568633 0.73 PADI4 (0.30) PADI4
SCHEMBL31488134 0.72 PADI4 (0.42) ADORA3ADORA1ADORA2APADI4
SCHEMBL24797436 0.63 PTGS2 (0.51)
SCHEMBL9876641 0.59 CDK4 (0.54) CYP2D6
SCHEMBL5370441 0.56 PKM (0.44) ADORA1ADORA2APIM1PIM2
SCHEMBL19007909 0.56 L3MBTL1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022140428-A2 INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2022-06-30 WO disclosed