SCHEMBL2465632

SCHEMBL2465632

C[Si](C)(C)C#Cc1ccc(NC(=O)O)c([N+](=O)[O-])c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
RAB9A P51151 8/20 0.43
NPC1 O15118 7/20 0.43
SMN1; SMN2 Q16637 5/20 0.43
MAPT P10636 5/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HCAR3 P49019 2/20 0.42
MAPK1 P28482 3/20 0.41
HTT P42858 2/20 0.41
GLA P06280 1/20 0.41
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
KMT2A Q03164 2/20 0.41
KCNMA1 Q12791 1/20 0.41
GAA P10253 1/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2465627 1.00 ALDH1A1 (0.45) ALDH1A1RAB9ANPC1SMN1; SMN2MAPT
SCHEMBL2133252 0.83 ADRA2A (0.41) ALDH1A1RAB9ANPC1SMN1; SMN2MAPT
SCHEMBL22636823 0.79 MAPT (0.55) ALDH1A1RAB9AMAPTNPSR1HCAR3
SCHEMBL6609844 0.79 ALDH1A1 (0.47) ALDH1A1RAB9ANPC1SMN1; SMN2MAPT
SCHEMBL1507617 0.79 ALDH1A1 (0.49) ALDH1A1RAB9ANPC1SMN1; SMN2MAPT
SCHEMBL2465151 0.78 GABRA1 (0.36) ALDH1A1RAB9ANPC1SMN1; SMN2MAPT
SCHEMBL21753178 0.77 GABRA1 (0.37) ALDH1A1MAPTKMT2AGAAMEN1
SCHEMBL6510043 0.77 VCAM1 (0.39) ALDH1A1RAB9ANPC1SMN1; SMN2MAPT
SCHEMBL21753062 0.76 PDK1 (0.43) ALDH1A1RAB9ANPC1SMN1; SMN2MAPT
SCHEMBL1704376 0.75 ALDH1A1 (0.71) ALDH1A1RAB9ANPC1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367599-A1 INHIBITION OF HDAC2 TO PROMOTE MEMORY Massachusetts Institute of Technology (US) 2011-09-28 EP disclosed
WO-2010065117-A1 INHIBITION OF HDAC2 TO PROMOTE MEMORY MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2010-06-10 WO disclosed