SCHEMBL247482

SCHEMBL247482

CC(C(=O)NNc1ccccn1)c1ccc(Cl)nn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 8/20 0.51
SMN1; SMN2 Q16637 5/20 0.50
POLB P06746 1/20 0.45
ALDH1A1 P00352 3/20 0.44
FFAR2 O15552 1/20 0.43
LMNA P02545 4/20 0.41
KDM4E B2RXH2 4/20 0.41
HTT P42858 4/20 0.41
KMT2A Q03164 2/20 0.41
MAPT P10636 2/20 0.41
GFER P55789 2/20 0.41
ALPL P05186 1/20 0.41
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.39
P2RX7 Q99572 1/20 0.39
TDP1 Q9NUW8 2/20 0.39
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1550986 0.72 GAA (0.50) GAASMN1; SMN2POLBALDH1A1LMNA
SCHEMBL28591272 0.71 FFAR2 (0.77) GAAFFAR2LMNAKDM4EHTT
SCHEMBL27850895 0.70 GAA (0.54) GAASMN1; SMN2POLBALDH1A1LMNA
SCHEMBL10877982 0.69 POLB (0.56) GAASMN1; SMN2POLBALDH1A1LMNA
SCHEMBL2696350 0.69 AKR1C3 (0.43) GAASMN1; SMN2POLBALDH1A1LMNA
SCHEMBL27668109 0.69 GAA (0.55) GAASMN1; SMN2ALDH1A1LMNAKDM4E
SCHEMBL29076327 0.68 GAA (0.58) GAASMN1; SMN2ALDH1A1LMNAKDM4E
SCHEMBL5954013 0.68 LMNA (0.50) GAAALDH1A1LMNAHTTKMT2A
SCHEMBL28595254 0.68 GAA (1.00) GAASMN1; SMN2POLBALDH1A1LMNA
SCHEMBL3709832 0.68 GAA (0.55) GAASMN1; SMN2POLBALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130315895-A1 COMBINATION OF A cMET INHIBITOR AND AN ANTIBODY TO HGF AND/OR cMET TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-11-28 US disclosed
EP-2588107-A1 COMBINATION OF A cMET INHIBITOR AND AN ANTIBODY TO HGF AND/OR cMET Takeda Pharmaceutical Company Limited (JP) 2013-05-08 EP disclosed
US-8178534-B2 cMET inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-05-15 US disclosed
WO-2012003338-A1 COMBINATION OF A cMET INHIBITOR AND AN ANTIBODY TO HGF AND/OR cMET TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-01-05 WO disclosed
EP-2313407-A1 cMET INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2011-04-27 EP disclosed
US-20100063054-A1 cMET INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-03-11 US disclosed
WO-2010019899-A1 cMET INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130315895-A1 COMBINATION OF A cMET INHIBITOR AND AN ANTIBODY TO HGF AND/OR cMET HGF, MET, HGFAC GAA 773/4885SMN1; SMN2 2559/4885POLB 3170/4885
US-20100063054-A1 cMET INHIBITORS CEPT1, LCAT, GNMT GAA 482/4885SMN1; SMN2 4131/4885POLB 2449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.