SCHEMBL2477683

SCHEMBL2477683

O=C(O)[C@@H]1CCCN1C(=O)c1cc2ccccc2nc1O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TRPV1 Q8NER1 1/20 0.44
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
OGFRL1 Q5TC84 1/20 0.44
CYP1A2 P05177 1/20 0.43
CA2 P00918 1/20 0.43
DGAT1 O75907 2/20 0.42
ITGB3 P05106 1/20 0.42
ITGB1 P05556 1/20 0.42
ITGAV P06756 1/20 0.42
ITGA5 P08648 1/20 0.42
ITGA4 P13612 1/20 0.42
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3695108 0.82 OPRM1 (0.54) ALDH1A1SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL6990139 0.81 SCD5 (0.53)
SCHEMBL2475715 0.79 CNR2 (0.55) ALDH1A1SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL2477407 0.79 CNR2 (0.55) ALDH1A1SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL2479401 0.78 CNR1 (0.57) ALDH1A1SMN1; SMN2CA2DGAT1
SCHEMBL6990119 0.77 HSP90AA1 (0.48) HSP90AA1HSP90AB1
SCHEMBL19474986 0.76 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2CA2DGAT1ITGB3
SCHEMBL19474987 0.76 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2CA2DGAT1ITGB3
SCHEMBL6987311 0.76 FABP4 (0.45) HSP90AA1HSP90AB1
SCHEMBL6989431 0.76 HCRTR2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373674-A1 2-(N-SUBSTITUTED PIPERAZINYL) STEROID DERIVATIVES Université Laval (CA) 2011-10-12 EP disclosed
WO-2010060215-A1 2-(N-SUBSTITUTED PIPERAZINYL) STEROID DERIVATIVES UNIVERSITé LAVAL (CA) 2010-06-03 WO disclosed