SCHEMBL2484727

SCHEMBL2484727

NC(=O)c1c(-c2ccccc2)ccc(C(F)(F)F)c1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
KDM4E B2RXH2 2/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
BCAT2 O15382 2/20 0.42
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
SCN9A Q15858 5/20 0.37
PLK1 P53350 1/20 0.37
ERN1 O75460 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
LDHA P00338 1/20 0.36
DHODH Q02127 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
FFAR4 Q5NUL3 1/20 0.35
CSNK1E P49674 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6677946 0.81 BCAT2 (0.49) ALDH1A1HPGDKDM4ELMNATSHR
SCHEMBL29978674 0.81 BCAT2 (0.49) ALDH1A1HPGDKDM4ELMNATSHR
SCHEMBL27967445 0.78 BCAT2 (0.42) ALDH1A1HPGDKDM4ELMNATSHR
SCHEMBL29702020 0.78 ALDH1A1 (0.43) ALDH1A1HPGDAKR1C3AKR1C2PLK1
SCHEMBL28636307 0.77 ALDH1A1 (0.45) ALDH1A1HPGDAKR1C3AKR1C2PLK1
SCHEMBL3763563 0.75 FABP4 (0.43) ALDH1A1HPGDKDM4ELMNATSHR
SCHEMBL27920522 0.75 GLA (0.38) ALDH1A1HPGDKDM4ETSHR
SCHEMBL27630251 0.74 ALDH1A1 (0.40) ALDH1A1HPGDKDM4ELMNATSHR
SCHEMBL403135 0.73 AKR1C3 (0.55) BCAT2AKR1C3AKR1C2SCN9AERN1
SCHEMBL6677822 0.73 TAS2R14 (0.44) ALDH1A1HPGDTSHRAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2375904-A1 BIARYL CARBOXAMIDES Merck Sharp & Dohme Corp. (US) 2011-10-19 EP claimed
WO-2010077624-A1 BIARYL CARBOXAMIDES MERCK SHARP & DOHME CORP. (US) 2010-07-08 WO claimed
CN-112707837-B Preparation method of N-cyclopropylmethylaniline compound 长沙嘉桥生物科技有限公司 2022-07-19 CN disclosed
CN-112707837-A Preparation method of N-cyclopropylmethylaniline compound 长沙嘉桥生物科技有限公司 2021-04-27 CN disclosed