SCHEMBL665545

SCHEMBL665545

Cc1ccsc1C(C(N)=O)c1nccs1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.47
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
PPARG P37231 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
CTSA P10619 8/20 0.37
ALDH1A1 P00352 1/20 0.35
ADAM17 P78536 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KDM4A O75164 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
KDM2A Q9Y2K7 1/20 0.34
NAMPT P43490 1/20 0.33
ADRA1D P25100 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL667099 0.77 CTSA (0.46) NPC1RAB9ACTSAALDH1A1
SCHEMBL667812 0.77 CTSA (0.34) ALOX5NPC1RAB9APPARGNCOR2
SCHEMBL5585939 0.74 ALDH1A1 (0.43) NPC1RAB9ACTSAALDH1A1ADAM17
SCHEMBL662588 0.74 CTSA (0.40) NPC1RAB9ACTSAALDH1A1NAMPT
SCHEMBL30497676 0.72 NPC1 (0.46) NPC1RAB9ACTSAALDH1A1SMN1; SMN2
SCHEMBL1007892 0.72 ALDH1A1 (0.42) CTSAALDH1A1KDM4ESMN1; SMN2
SCHEMBL666602 0.71 CTSA (0.52) NPC1RAB9ACTSA
SCHEMBL27953126 0.71 ALOX5 (0.50) ALOX5NPC1RAB9APPARGNCOR2
SCHEMBL662300 0.71 CYP1A2 (0.41) CTSA
SCHEMBL12495359 0.70 GCK (0.38) CTSAALDH1A1KDM4EKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180133170-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS ELI LILLY AND COMPANY 2018-05-17 US disclosed
US-20130165427-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CHEMICAL WARFARE AGENT-INDUCED INJURIES HYDRA BIOSCIENCES, INC. (US) 2013-06-27 US disclosed
US-20130059869-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS HYDRA BIOSCIENCES, INC. 2013-03-07 US disclosed
US-20120108614-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CHEMICAL WARFARE AGENT-INDUCED INJURIES HYDRA BIOSCIENCES, INC. 2012-05-03 US disclosed
US-20120046305-A1 METHODS AND COMPOSITIONS FOR TREATING RESPIRATORY DISORDERS ELI LILLY AND COMPANY 2012-02-23 US disclosed
US-20090143377-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS ELI LILLY AND COMPANY 2009-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120108614-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CHEMICAL WARFARE AGENT-INDUCED INJURIES ELANE, CASP3, MMP8 ALOX5 1181/4885NPC1 2375/4885RAB9A 1580/4885
US-20180133170-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS TRPA1, TRPV1, TRPV3 ALOX5 138/4885NPC1 73/4885RAB9A 2306/4885
US-20090143377-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS TRPA1, TRPV1, TRPV3 ALOX5 138/4885NPC1 73/4885RAB9A 2306/4885
US-20120046305-A1 METHODS AND COMPOSITIONS FOR TREATING RESPIRATORY DISORDERS TRPA1, TRPV1, TRPV3 ALOX5 212/4885NPC1 283/4885RAB9A 2725/4885
US-20130165427-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CHEMICAL WARFARE AGENT-INDUCED INJURIES ELANE, CASP3, MMP8 ALOX5 1181/4885NPC1 2375/4885RAB9A 1580/4885
US-20130059869-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS TRPA1, TRPV1, TRPV3 ALOX5 138/4885NPC1 73/4885RAB9A 2306/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.