SCHEMBL253706

SCHEMBL253706

O=C(NCc1cccc(C(F)(F)F)c1)c1cnc2ncccc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.58
PSMD14 O00487 4/20 0.58
STAMBP O95630 3/20 0.58
CYP3A4 P08684 2/20 0.57
CYP2C19 P33261 2/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
PLA2G1B P04054 1/20 0.57
CYP1A2 P05177 1/20 0.57
GAA P10253 1/20 0.57
CYP2D6 P10635 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
ATG4B Q9Y4P1 1/20 0.57
DHFR P00374 1/20 0.55
CYP2C9 P11712 1/20 0.54
NAMPT P43490 1/20 0.54
HDAC3 O15379 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13491609 0.83 MLYCD (0.62) MLYCDCYP3A4CYP2C19MEN1KMT2A
SCHEMBL247656 0.83 LMNA (0.54) MLYCDCYP3A4CYP2C19MEN1KMT2A
SCHEMBL247884 0.81 LMNA (0.52) MLYCDCYP3A4CYP2C19MEN1KMT2A
SCHEMBL616941 0.81 DHFR (0.56) MLYCDCYP3A4CYP2C19MEN1KMT2A
SCHEMBL619841 0.80 LMNA (0.51) MLYCDCYP3A4CYP2C19MEN1KMT2A
SCHEMBL5697540 0.80 PSMD14 (0.54) PSMD14STAMBPCYP3A4MAPK14ROCK2
SCHEMBL252287 0.79 STAMBP (0.51) PSMD14STAMBPCYP3A4CYP2C19CYP2C9
SCHEMBL619692 0.79 RIPK1 (0.51) MLYCDCYP3A4CYP2C19MEN1KMT2A
SCHEMBL253234 0.78 PSMD14 (0.50) PSMD14STAMBPCYP3A4CYP2C19CYP1A2
SCHEMBL1568282 0.78 MLYCD (0.74) MLYCDCYP3A4CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP claimed
EP-2401275-B1 NAPHTHYRIDINE DERIVATIVES HAVING BRONCHODILATING ACTIVITY RESPIRATORIUS AB (SE) 2013-07-24 EP disclosed
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP disclosed