SCHEMBL25519458

SCHEMBL25519458

Cc1cc(C#N)ccc1-c1nnc(N)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 6/20 0.41
HSP90AB1 P08238 1/20 0.39
NSD2 O96028 2/20 0.36
AR P10275 5/20 0.36
TRPV4 Q9HBA0 1/20 0.36
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
KIF11 P52732 1/20 0.35
SLC22A12 Q96S37 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25519495 0.83 EGLN2 (0.46) EGLN2HSP90AB1NSD2CYP11B1CYP11B2
SCHEMBL3366225 0.77 HSP90AB1 (0.44) EGLN2HSP90AB1NSD2CYP11B1CYP11B2
SCHEMBL25519380 0.72 NLRP3 (0.50) EGLN2HSP90AB1NSD2CYP11B1CYP11B2
SCHEMBL3399428 0.72 CYP11B1 (0.39) EGLN2NSD2TRPV4CYP11B1CYP11B2
SCHEMBL171819 0.71 KIF11 (0.51) ARTRPV4KIF11SLC22A12
SCHEMBL23770666 0.71 KRAS (0.39) EGLN2NSD2ARTRPV4CYP11B1
SCHEMBL20116875 0.69 ALDH1A1 (0.45) EGLN2ARCYP11B1CYP11B2SLC22A12
SCHEMBL2154193 0.69 CYP11B2 (0.53) EGLN2ARCYP11B1CYP11B2SLC22A12
SCHEMBL409405 0.68 TRPV4 (0.53) ARTRPV4KIF11
SCHEMBL7604551 0.68 TRPV4 (0.56) NSD2ARTRPV4KIF11SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023088987-A1 PYRIDAZINE DERIVATIVES AS INHIBITORS OF NLRP3 F. HOFFMANN-LA ROCHE AG (CH) 2023-05-25 WO disclosed