SCHEMBL25519495

SCHEMBL25519495

Cc1cc(C#N)ccc1-c1nnc(N)cc1C

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 6/20 0.46
CYP11B2 P19099 6/20 0.40
CYP11B1 P15538 5/20 0.40
HSP90AB1 P08238 1/20 0.40
NLRP3 Q96P20 3/20 0.39
NSD2 O96028 2/20 0.38
KCNH2 Q12809 1/20 0.36
SLC22A12 Q96S37 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25519380 0.88 NLRP3 (0.50) EGLN2CYP11B2CYP11B1HSP90AB1NLRP3
SCHEMBL25519458 0.83 EGLN2 (0.41) EGLN2CYP11B2CYP11B1HSP90AB1NSD2
SCHEMBL20116875 0.76 ALDH1A1 (0.45) EGLN2CYP11B2CYP11B1SLC22A12
SCHEMBL2154193 0.75 CYP11B2 (0.53) EGLN2CYP11B2CYP11B1SLC22A12
SCHEMBL25856432 0.73 NLRP3 (0.38) NLRP3
SCHEMBL3364120 0.73 EGLN2 (0.47) EGLN2CYP11B2CYP11B1HSP90AB1NSD2
SCHEMBL25859518 0.72 NLRP3 (0.37) NLRP3
SCHEMBL3366217 0.71 KCNH2 (0.52) EGLN2CYP11B2CYP11B1KCNH2
SCHEMBL17630059 0.71 EGLN2 (0.47) EGLN2CYP11B2CYP11B1HSP90AB1NSD2
SCHEMBL25856428 0.71 NLRP3 (0.36) NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023088987-A1 PYRIDAZINE DERIVATIVES AS INHIBITORS OF NLRP3 F. HOFFMANN-LA ROCHE AG (CH) 2023-05-25 WO disclosed