SCHEMBL2555945

SCHEMBL2555945

COC(=O)c1cccc2c1NC(c1cccc(C(=O)N(C)C3CCNC3)c1)C(C)(C)C2

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 18/20 0.43
SLC6A2 P23975 17/20 0.43
KCNH2 Q12809 6/20 0.43
SLC6A3 Q01959 10/20 0.35
BTK Q06187 1/20 0.34
CYP2D6 P10635 3/20 0.33
MCHR1 Q99705 1/20 0.33
OPRK1 P41145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2591486 0.91 SLC6A4 (0.45) SLC6A4SLC6A2KCNH2SLC6A3BTK
SCHEMBL2533630 0.81 KMO (0.37) SLC6A3
SCHEMBL2582189 0.77 CHRNB2 (0.40)
SCHEMBL2531549 0.74 RAB9A (0.45) SLC6A2SLC6A3
SCHEMBL2531741 0.73 ROCK2 (0.40) MCHR1
SCHEMBL11026198 0.69 ALDH1A1 (0.39)
SCHEMBL2535744 0.68 ADRA1D (0.41)
SCHEMBL3065694 0.67 SLC6A4 (0.62) SLC6A4SLC6A2KCNH2SLC6A3CYP2D6
SCHEMBL3065696 0.67 SLC6A4 (0.62) SLC6A4SLC6A2KCNH2SLC6A3CYP2D6
SCHEMBL27888392 0.67 GAA (0.41) SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed