SCHEMBL25614129

SCHEMBL25614129

Brc1cncc(-n2cccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 7/20 0.44
CHRNA4 P43681 7/20 0.44
CHRNB4 P30926 5/20 0.44
CHRNA3 P32297 5/20 0.44
POLB P06746 2/20 0.36
HCAR2 Q8TDS4 1/20 0.36
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
MAPT P10636 1/20 0.33
CYP2A6 P11509 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PTK2 Q05397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30811828 1.00 CHRNB2 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3POLB
SCHEMBL1502674 0.78 CHRNB2 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3POLB
SCHEMBL1559218 0.78 CYP3A4 (0.52) CHRNB2CHRNA4ALOX15MAPTCYP2A6
SCHEMBL5659919 0.74 CHRNB2 (0.47) CHRNB2CHRNA4CHRNB4CHRNA3POLB
SCHEMBL30201408 0.74 MAPT (0.52) POLBMAPTCYP2A6KDM4EMEN1
SCHEMBL16720482 0.74 CHRNB2 (0.42) CHRNB2CHRNA4POLBMAPTCYP2A6
SCHEMBL3931376 0.74 MAPT (0.52) POLBMAPTCYP2A6KDM4EMEN1
SCHEMBL12369610 0.74 CHRNB2 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3POLB
SCHEMBL14909303 0.74 HTT (0.40) CHRNB2CHRNA4CHRNB4CHRNA3POLB
SCHEMBL30811728 0.72 CHRNB2 (0.56) CHRNB2CHRNA4CHRNB4CHRNA3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4582422-A1 METTL3 INHIBITOR COMPOUND, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF Global Health Drug Discovery Institute (CN) 2025-07-09 EP disclosed
US-20250214997-A1 METTL3 INHIBITOR COMPOUND, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF GLOBAL HEALTH DRUG DISCOVERY INSTITUTE (CN) 2025-07-03 US disclosed
CN-117736182-A MetTL3 inhibitors and uses thereof 成都先导药物开发股份有限公司 2024-03-22 CN disclosed
WO-2024056099-A1 METTL3 INHIBITOR COMPOUND, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 北京华益健康药物研究中心 2024-03-21 WO disclosed
US-11802120-B2 Fused cyclic urea derivatives as CRHR2 antagonist RAQUALIA PHARMA INC. (JP) 2023-10-31 US disclosed
WO-2023104209-A1 METTL3 INHIBITOR COMPOUND 上海昂阔医药有限公司 2023-06-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11802120-B2 Fused cyclic urea derivatives as CRHR2 antagonist CRHR2, CRHR1, CRH CHRNB2 1703/4885CHRNA4 2400/4885CHRNB4 2651/4885
US-20250214997-A1 METTL3 INHIBITOR COMPOUND, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF METTL3, METTL14, METTL16 CHRNB2 4468/4885CHRNA4 4400/4885CHRNB4 4350/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.