SCHEMBL257644

SCHEMBL257644

Bc1cc(F)c(C(=O)O)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA4 P22748 3/20 0.34
RARA P10276 2/20 0.34
RARG P13631 2/20 0.34
RARB P10826 1/20 0.34
KDM4E B2RXH2 4/20 0.33
ASPH Q12797 1/20 0.33
KDM8 Q8N371 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
HSD17B10 Q99714 3/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HCAR1 Q9BXC0 1/20 0.32
NOTUM Q6P988 1/20 0.32
CYP1A2 P05177 1/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21000330 0.85 CYP3A4 (0.42) KDM4EHSD17B10ALDH1A1HPGDMEN1
SCHEMBL19220334 0.84 RARA (0.32) CA1CA2CA4RARARARG
SCHEMBL28888036 0.79 AKR1C2 (0.45) CA1CA2CA4RARARARG
SCHEMBL288979 0.79 CES2 (0.46) CA1CA2CA4RARARARG
SCHEMBL28267100 0.78 DGAT1 (0.41) CA1CA2CA4CES2CES1
SCHEMBL17177745 0.77 AKR1C2 (0.44) CA1CA2CA4RARARARG
SCHEMBL198786 0.77 HCAR1 (0.48) CA1CA2CA4RARARARG
SCHEMBL542833 0.77 LMNA (0.50) CA1CA2CA4KDM4EHSD17B10
SCHEMBL29154306 0.77 CES2 (0.44) CA1CA2CA4RARARARG
SCHEMBL7567840 0.75 CA1 (0.56) CA1CA2CA4KDM4EASPH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3042903-B1 Substituted hetero-bicyclic compounds, compositions and medicinal applications thereof IMPETIS BIOSCIENCES LTD (IN) 2019-08-14 EP disclosed
WO-2012029942-A1 CYCLIC AMIDE DERIVATIVE 大日本住友製薬株式会社 (JP) 2012-03-08 WO disclosed