SCHEMBL2578770

SCHEMBL2578770

CCOC(=O)C(C)NC(=O)c1noc2c1CN(C(=O)c1ccc(OC)cc1)CC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 10/20 0.48
MAPT P10636 4/20 0.43
TSHR P16473 2/20 0.43
RAB9A P51151 3/20 0.43
ATM Q13315 1/20 0.43
NPC1 O15118 2/20 0.43
RECQL P46063 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
NR4A1 P22736 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GAA P10253 1/20 0.42
LMNA P02545 3/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2578771 0.83 HSP90AA1 (0.49) HSP90AA1MAPTTSHRRAB9AATM
SCHEMBL4259746 0.80 LMNA (0.50) HSP90AA1MAPTTSHRRAB9ANPC1
SCHEMBL2582339 0.79 HSP90AA1 (0.49) HSP90AA1MAPTTSHRRAB9AATM
SCHEMBL5527334 0.72 HPGD (0.46) MAPTTSHRNPC1ALDH1A1POLB
SCHEMBL2585252 0.72 PKM (0.46) HSP90AA1MAPTTSHRRAB9ANPC1
SCHEMBL2578696 0.71 SMN1; SMN2 (0.66) MAPTTSHRRAB9AATMNPC1
SCHEMBL2582491 0.70 ALDH1A1 (0.48) MAPTTSHRRAB9AATMNPC1
SCHEMBL2582494 0.68 KMT2A (0.44) HSP90AA1MAPTTSHRRAB9AATM
SCHEMBL12487063 0.68 RAB9A (0.42) HSP90AA1MAPTTSHRRAB9AATM
SCHEMBL12487066 0.68 RAB9A (0.42) HSP90AA1MAPTTSHRRAB9AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US claimed