SCHEMBL25832

SCHEMBL25832

NC(=O)C12CCC(CC(NS(=O)(=O)c3ccc(Oc4ccc(Cl)cc4)cc3)(C(=O)O)C1)O2

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 16/20 0.57
MMP13 P45452 16/20 0.57
MMP2 P08253 3/20 0.46
MMP9 P14780 3/20 0.46
MMP3 P08254 2/20 0.46
MMP8 P22894 2/20 0.46
ADAMTS5 Q9UNA0 2/20 0.40
USP2 O75604 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MMP12 P39900 1/20 0.39
MMP14 P50281 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25908 0.92 MMP1 (0.56) MMP1MMP13MMP2MMP9MMP3
SCHEMBL4575861 0.79 MMP1 (0.42) MMP1MMP13MMP2MMP9MMP3
SCHEMBL27450137 0.78 MMP1 (0.65) MMP1MMP13MMP2MMP9MMP3
Hydroxyamine SCHEMBL7514521 0.75 MMP1 (0.76) MMP1MMP13MMP2MMP9MMP3
SCHEMBL12076423 0.75 MMP1 (0.79) MMP1MMP13MMP2MMP9MMP3
SCHEMBL250645 0.74 MMP1 (0.76) MMP1MMP13MMP2MMP9MMP3
Hydroxyamine SCHEMBL3874403 0.74 MMP1 (0.77) MMP1MMP13MMP2MMP9MMP3
SCHEMBL3667056 0.74 MMP1 (0.80) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7214294 0.73 MMP1 (0.80) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7209172 0.73 MMP1 (0.80) MMP1MMP13MMP2MMP9MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 530 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534153-B2 SALTS AND POLYMORPHS OF 8-FLUORO-2-{4-[(METHYLAMINO}METHYL]PHENYL}-1,3,4,5-TETRAHYDRO-6H-AZEPINO[5,4,3-CD]INDOL-6-ONE PFIZER (US) 2024-05-22 EP disclosed
US-20240109862-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER INC. 2024-04-04 US disclosed
EP-3590932-B1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE SUMITOMO PHARMA ONCOLOGY INC (US) 2023-05-03 EP disclosed
EP-4166558-A1 SALTS AND POLYMORPHS OF 8-FLUORO-2-{4- [(METHYLAMINO)METHYL]PHENYL}-1 ,3,4,5-TETRAHYDRO-6H-AZEPINO[5,4,3- CD]INDOL-6-ONE Pfizer Inc. (US) 2023-04-19 EP disclosed
US-20220162200-A1 PKM2 MODULATORS AND METHODS FOR THEIR USE SUMITOMO DAINIPPON PHARMA ONCOLOGY, INC. 2022-05-26 US disclosed
US-11124499-B2 Pharmaceutical composition derived from Tecoma plant and a method for treating cancer NATIONAL GUARD HEALTH AFFAIRS (SA) 2021-09-21 US disclosed
US-20210277037-A1 DEUTERATED ALVOCIDIB AND ALVOCIDIB PRODRUGS SUMITOMO PHARMA ONCOLOGY, INC. 2021-09-09 US disclosed
US-20210238183-A1 SUBSTITUTED IMIDAZO[1,2-B]PYRIDAZINES AS PROTEIN KINASE INHIBITORS SUMITOMO PHARMA AMERICA, INC. 2021-08-05 US disclosed
EP-3812387-A1 HETEROCYCLIC PROTEIN KINASE INHIBITORS Sumitomo Dainippon Pharma Oncology, Inc. (US) 2021-04-28 EP disclosed
US-20210070715-A1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE SUMITOMO PHARMA AMERICA, INC. 2021-03-11 US disclosed
US-20020019530-A1 Heteroaryl-substituted quinolin-2-one derivatives useful as anticancer agents YANG BINGWEI V (US) 2002-02-14 US disclosed
WO-2002010141-A1 IMIDAZOLE DERIVATIVES PFIZER PRODUCTS INC. (US) 2002-02-07 WO disclosed
EP-1177791-A2 Use of glycogen phosphorylase inhibitors to inhibit tumor growth Pfizer Products Inc. (US) 2002-02-06 EP disclosed
US-20020004511-A1 Thiophene derivatives useful as anticancer agents LUZZIO MICHAEL JOSEPH (US) 2002-01-10 US disclosed
WO-2001098277-A2 SUBSTITUTED BICYCLIC DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER PRODUCTS INC. (US) 2001-12-27 WO disclosed
WO-2001094353-A1 THIOPHENE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 2001-12-13 WO disclosed
WO-2001053289-A1 ANTICANCER COMPOUND AND ENANTIOMER SEPARATION METHOD USEFUL FOR SYNTHESIZING SAID COMPOUND PFIZER PRODUCTS INC. (US) 2001-07-26 WO disclosed
US-6258824-B1 TREATMENT OF HYPERPROLIFERATIVE DISEASES, SUCH AS CANCERS, IN MAMMALS. THIS INVENTION ALSO RELATES TO A PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDS. PFIZER INC. 2001-07-10 US disclosed
EP-1106612-A1 Quinoline derivatives useful for inhibiting farnesyl protein transferase Pfizer Products Inc. (US) 2001-06-13 EP disclosed
WO-2001040217-A1 NOVEL BENZOIMIDAZOLE DERIVATIVES USEFUL AS ANTIPROLIFERATIVE AGENTS PFIZER PRODUCTS INC. (US) 2001-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020004511-A1 Thiophene derivatives useful as anticancer agents CCNA1, CCNE1, TP53 MMP1 2429/4885MMP13 4017/4885MMP2 4517/4885
US-20210070715-A1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE ALK, JAK2, JAK1 MMP1 2298/4885MMP13 2440/4885MMP2 2512/4885
US-20220162200-A1 PKM2 MODULATORS AND METHODS FOR THEIR USE PDK1, PKM, PDK2 MMP1 4359/4885MMP13 3911/4885MMP2 3348/4885
US-20210238183-A1 SUBSTITUTED IMIDAZO[1,2-B]PYRIDAZINES AS PROTEIN KINASE INHIBITORS PIM1, PIM2, PIM3 MMP1 2061/4885MMP13 4280/4885MMP2 3813/4885
US-20210277037-A1 DEUTERATED ALVOCIDIB AND ALVOCIDIB PRODRUGS CDK4, CDK11B, CDK3 MMP1 1315/4885MMP13 820/4885MMP2 1970/4885
US-20020019530-A1 Heteroaryl-substituted quinolin-2-one derivatives useful as anticancer agents NRAS, CCNA1, KRAS MMP1 4314/4885MMP13 3790/4885MMP2 3550/4885
US-20240109862-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH GPR119, INSR, LYAR MMP1 3955/4885MMP13 4604/4885MMP2 4086/4885
US-11124499-B2 Pharmaceutical composition derived from Tecoma plant and a method for treating cancer TEC, TMSB10, MALT1 MMP1 3159/4885MMP13 931/4885MMP2 2546/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.