SCHEMBL25858995

SCHEMBL25858995

CC#Cc1ccc(-c2nnc(NC)nc2C)c(O)c1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.38
EGLN1 Q9GZT9 1/20 0.32
HSD17B10 Q99714 1/20 0.31
CYP1A1 P04798 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP1B1 Q16678 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25861616 0.85 NLRP3 (0.39) NLRP3HSD17B10
SCHEMBL25857850 0.77 NLRP3 (0.42) NLRP3EGLN1
SCHEMBL25856264 0.76 IL1B (0.51) NLRP3
SCHEMBL25857462 0.75 NLRP3 (0.62) NLRP3
SCHEMBL25861920 0.75 NLRP3 (0.39) NLRP3HSD17B10
SCHEMBL25858838 0.73 ALDH1A1 (0.45) NLRP3CYP1A1CYP1A2CYP1B1
SCHEMBL25859518 0.71 NLRP3 (0.37) NLRP3EGLN1
SCHEMBL25858377 0.70 NLRP3 (0.35) NLRP3
SCHEMBL25860307 0.69 EGFR (0.31)
SCHEMBL25860146 0.69 NLRP3 (0.31) NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed