SCHEMBL260254

SCHEMBL260254

CC(O)C(=O)OC(C)C(=O)OCC(=O)OCC(=O)O

nearest known ligand 0.37

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PAM P19021 3/20 0.37
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14866116 0.95 PAM (0.34) PAM
SCHEMBL4261273 0.87 PAM (0.42) PAMTP53
SCHEMBL13949509 0.86
SCHEMBL18162008 0.85 PAM (0.41) PAM
SCHEMBL15504792 0.84
SCHEMBL13949506 0.79
SCHEMBL41709 0.78 TP53 (0.43) PAMTP53
SCHEMBL27483337 0.78 TP53 (0.43) PAMTP53
SCHEMBL18159124 0.78 NAAA (0.49) PAM
SCHEMBL17368711 0.78 NAAA (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170354592-A1 PARENTERAL SUSTAINED-RELEASE DELIVERY OF CARVEDILOL DISPERSE SYSTEMS ASCENDIA PHARMACEUTICALS, LLC (US) 2017-12-14 US disclosed
US-20140377369-A2 COMPOSITIONS OF ROTIGOTINE, DERIVATIVES THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS OF ROTIGOTINE OR ITS DERIVATIVES GENEORA PHARMA (SHIJIAZHUANG) CO., LTD. (CN) 2014-12-25 US disclosed
US-20130309314-A1 COMPOSITIONS OF ROTIGOTINE, DERIVATIVES THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS OF ROTIGOTINE OR ITS DERIVATIVE LI YOUXIN (DE) 2013-11-21 US disclosed
US-8481558-B2 Compounds to inhibit or augment an inflammatory response CAMBRIDGE ENTERPRISE LIMITED (GB) 2013-07-09 US disclosed
US-20120065401-A1 METHODS TO INHIBIT OR AUGMENT AN INFLAMMATORY RESPONSE CAMBRIDGE ENTERPRISE LIMITED (GB) 2012-03-15 US disclosed
US-8067022-B2 Inhibiting stenosis following vascular trauma or disease by administering a conjugate of a vascular smooth muscle binding protein that associates with a cell surface of the vascular smooth muscle coupled to a drug inhibiting cellular activity BOSTON SCIENTIFIC SCIMED, INC. (US) 2011-11-29 US disclosed
US-7989466-B2 Administering chemokine peptides, variants, and derivatives thereof, as well as chemokine peptide analogs to modulate the migration or recruitment of leukocytes to a preselected physiological site CAMBRIDGE ENTERPRISE LIMITED (GB) 2011-08-02 US disclosed
US-20090196931-A1 THERAPEUTIC INHIBITOR OF VASCULAR SMOOTH MUSCLE CELLS KUNZ LAWRENCE L 2009-08-06 US disclosed
US-20080045557-A1 Administering chemokine peptides, variants, and derivatives thereof, as well as chemokine peptide analogs to modulate the migration or recruitment of leukocytes to a preselected physiological site CAMBRIDGE UNIVERSITY TECHNICAL SERVICES LTD. 2008-02-21 US disclosed
US-7238711-B1 Compounds and methods to inhibit or augment an inflammatory response CAMBRIDGE UNIVERSITY TECHNICAL SERVICES LTD. (GB) 2007-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130309314-A1 COMPOSITIONS OF ROTIGOTINE, DERIVATIVES THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS OF ROTIGOTINE OR ITS DERIVATIVE PARK7, PRLHR, PRPH PAM 2907/4885TP53 4538/4885
US-20090196931-A1 THERAPEUTIC INHIBITOR OF VASCULAR SMOOTH MUSCLE CELLS MYLK, TNNI3, MYLK2 PAM 3818/4885TP53 4453/4885
US-20140377369-A2 COMPOSITIONS OF ROTIGOTINE, DERIVATIVES THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS OF ROTIGOTINE OR ITS DERIVATIVES PARK7, PRLHR, ADCYAP1R1 PAM 2997/4885TP53 4638/4885
US-20080045557-A1 Administering chemokine peptides, variants, and derivatives thereof, as well as chemokine peptide analogs to modulate the migration or recruitment of leukocytes to a preselected physiological site CCL2, CCL11, CCL5 PAM 3543/4885TP53 2268/4885
US-20170354592-A1 PARENTERAL SUSTAINED-RELEASE DELIVERY OF CARVEDILOL DISPERSE SYSTEMS NPC1L1, PNLIP, LIPA PAM 4254/4885TP53 4672/4885
US-20120065401-A1 METHODS TO INHIBIT OR AUGMENT AN INFLAMMATORY RESPONSE CCL2, CCL5, CCL11 PAM 3306/4885TP53 2219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.