Methopholine

Methopholine

SCHEMBL26169

COc1cc2c(cc1OC)C(CCc1ccc(Cl)cc1)N(C)CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 1.00
MAOA P21397 1/20 1.00
PTGS2 P35354 1/20 1.00
OPRK1 P41145 1/20 1.00
SLC6A3 Q01959 1/20 1.00
MAPK1 P28482 2/20 0.82
TP53 P04637 1/20 0.82
TSHR P16473 1/20 0.82
KCNN2 Q9H2S1 4/20 0.67
KCNN3 Q9UGI6 4/20 0.67
KCNN1 Q92952 2/20 0.67
LMNA P02545 2/20 0.65
KDM4E B2RXH2 2/20 0.65
ALDH1A1 P00352 2/20 0.65
HSD17B10 Q99714 2/20 0.65
CYP2D6 P10635 1/20 0.65
GRIN2D O15399 4/20 0.64
GRIN3B O60391 4/20 0.64
GRIN1 Q05586 4/20 0.64
GRIN2A Q12879 4/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methopholine SCHEMBL30492235 1.00 NR1I2 (1.00) NR1I2MAOAPTGS2OPRK1SLC6A3
SCHEMBL29651290 0.91 TP53 (0.98) NR1I2MAOAPTGS2OPRK1SLC6A3
SCHEMBL5908036 0.91 TP53 (0.98) NR1I2MAOAPTGS2OPRK1SLC6A3
Hydrochloric Acid SCHEMBL2000082 0.90 TP53 (1.00) NR1I2MAOAPTGS2OPRK1SLC6A3
SCHEMBL8203917 0.89 NR1I2 (0.80) NR1I2MAOAPTGS2OPRK1SLC6A3
SCHEMBL27961570 0.84 MAOA (0.72) NR1I2MAOAPTGS2OPRK1SLC6A3
SCHEMBL8200503 0.83 TP53 (0.78) NR1I2MAOAPTGS2OPRK1SLC6A3
SCHEMBL3253219 0.81 KCNN2 (0.94) NR1I2MAOAPTGS2OPRK1SLC6A3
SCHEMBL3250242 0.81 KCNN2 (1.00) NR1I2MAOAPTGS2OPRK1SLC6A3
Homolaudanosine SCHEMBL7550998 0.80 NR1I2 (0.67) NR1I2MAOAPTGS2OPRK1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1491 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3560484-A1 ABUSE-DETERRENT PHARMACEUTICAL COMPOSITION G.L. Pharma GmbH (AT) 2019-10-30 EP claimed
EP-3423034-B1 ABUSE-DETERRENT PHARMACEUTICAL COMPOSITION G L PHARMA GMBH (AT) 2019-07-10 EP claimed
EP-3423034-A1 ABUSE-DETERRENT PHARMACEUTICAL COMPOSITION G.L. Pharma GmbH (AT) 2019-01-09 EP claimed
CN-109069419-A Abuse resistant drugs composition G.L.制药有限责任公司 2018-12-21 CN claimed
EP-3210596-A1 ABUSE-DETERRENT PHARMACEUTICAL COMPOSITION G.L. Pharma GmbH (AT) 2017-08-30 EP claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-20120063996-A1 NOVEL NIMESULIDE COMPOSITIONS ELAN PHARMA INTERNATIONAL LTD. 2012-03-15 US claimed
EP-1617816-B1 NANOPARTICULATE MELOXICAN FORMULATIONS ELAN PHARMA INT LTD (IE) 2009-05-13 EP claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
US-20040156872-A1 Novel nimesulide compositions ELAN PHARMA INTERNATIONAL LTD. 2004-08-12 US claimed
US-20040105881-A1 Aggregates with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2004-06-03 US claimed
WO-2004032900-A1 AGGREGATE WITH INCREASED DEFORMABILITY, COMPRISING AT LEAST THREE AMPHIPATS, FOR IMPROVED TRANSPORT THROUGH SEMI-PERMEABLE BARRIERS AND FOR THE NON-INVASIVE DRUG APPLICATION IN VIVO, ESPECIALLY THROUGH THE SKIN IDEA AG (DE) 2004-04-22 WO claimed
US-20030235617-A1 Pharmaceutical dosage form for mucosal delivery MCNEIL-PPC, INC 2003-12-25 US claimed
US-20030180357-A1 Pharmaceutical tablet MCNEIL-PPC, INC 2003-09-25 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
WO-2003066029-A2 PHARMACEUTICAL DOSAGE FORM FOR MUCOSAL DELIVERY PHARMACIA CORPORATION (US) 2003-08-14 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040156872-A1 Novel nimesulide compositions NIM1K, NIT2, NCL NR1I2 3919/4885MAOA 277/4885PTGS2 2387/4885
US-20030180357-A1 Pharmaceutical tablet GYPA, SORD, SRI NR1I2 1613/4885MAOA 1137/4885PTGS2 593/4885
US-20120063996-A1 NOVEL NIMESULIDE COMPOSITIONS NIM1K, NIT2, NCL NR1I2 3919/4885MAOA 277/4885PTGS2 2387/4885
US-20040105881-A1 Aggregates with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin CUTA, ABCG2, PIGS NR1I2 1134/4885MAOA 2457/4885PTGS2 2551/4885
US-20030235617-A1 Pharmaceutical dosage form for mucosal delivery SI, UGGT1, GYPA NR1I2 1375/4885MAOA 1023/4885PTGS2 557/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.