SCHEMBL26217525

SCHEMBL26217525

CCN(CC(=O)N(C)c1ccc(OC)cc1)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.43
HSD17B2 P37059 2/20 0.43
MTNR1A P48039 4/20 0.41
MTNR1B P49286 4/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
CETP P11597 2/20 0.40
LMNA P02545 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.40
KMT2A Q03164 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26222015 0.89 HSD17B1 (0.41) HSD17B1HSD17B2MTNR1AMTNR1BNPC1
SCHEMBL26217412 0.83 BCL2A1 (0.47) HSD17B1HSD17B2MAPTTP53POLB
SCHEMBL26217384 0.82 LMNA (0.51) MTNR1AMTNR1BNPC1RAB9AMAPT
SCHEMBL26217468 0.82 ALDH1A1 (0.47) NPC1RAB9AMAPTTP53POLB
SCHEMBL26217430 0.78 CETP (0.43) MAPTTP53POLBCETPLMNA
SCHEMBL26217555 0.78 L3MBTL1 (0.48) RAB9AMAPTLMNAMEN1ALDH1A1
SCHEMBL26221117 0.76 POLQ (0.45) NPC1RAB9AMAPTTP53POLB
SCHEMBL26217594 0.76 ALDH1A1 (0.46) NPC1RAB9AMAPTTP53POLB
SCHEMBL26217450 0.73 LMNA (0.45) NPC1RAB9AMAPTTP53POLB
SCHEMBL26217487 0.73 LMNA (0.45) NPC1RAB9AMAPTTP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230399292-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS PTC Innovations, LLC 2023-12-14 US disclosed
US-20230399291-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS PTC INNOVATIONS LLC (US) 2023-12-14 US disclosed
US-20230399290-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS PTC INNOVATIONS LLC (US) 2023-12-14 US disclosed
US-20230373906-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS PTC INNOVATIONS LLC (US) 2023-11-23 US disclosed
US-11814335-B1 Anesthetic compounds and methods of making and using same to treat or prevent pain symptoms PTC Innovations, LLC (US) 2023-11-14 US disclosed
US-11786493-B2 Anesthetic compounds and methods of making and using same to treat or prevent pain symptoms PTC Innovations, LLC (US) 2023-10-17 US disclosed
WO-2023172603-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS PTC Innovations, LLC (US) 2023-09-14 WO disclosed
US-20230286905-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS PTC Innovations, LLC 2023-09-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230399290-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS OPRK1, ACHE, F5 HSD17B1 1645/4885HSD17B2 1193/4885MTNR1A 1840/4885
US-20230399292-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS OPRM1, OPRL1, OPRK1 HSD17B1 2498/4885HSD17B2 2269/4885MTNR1A 40/4885
US-20230399291-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS CHRM2, RXFP2, OPRM1 HSD17B1 3392/4885HSD17B2 2028/4885MTNR1A 242/4885
US-11814335-B1 Anesthetic compounds and methods of making and using same to treat or prevent pain symptoms F8, F5, OPRM1 HSD17B1 1484/4885HSD17B2 1078/4885MTNR1A 1935/4885
US-20230286905-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS OPRM1, OPRL1, OPRK1 HSD17B1 1401/4885HSD17B2 1434/4885MTNR1A 55/4885
US-20230373906-A1 ANESTHETIC COMPOUNDS AND METHODS OF MAKING AND USING SAME TO TREAT OR PREVENT PAIN SYMPTOMS F5, EIF4G2, ACHE HSD17B1 1272/4885HSD17B2 857/4885MTNR1A 1187/4885
US-11786493-B2 Anesthetic compounds and methods of making and using same to treat or prevent pain symptoms OPRM1, OPRL1, OPRK1 HSD17B1 1401/4885HSD17B2 1434/4885MTNR1A 55/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.