SCHEMBL26459262

SCHEMBL26459262

CS(=O)(=O)c1cc(O)c2c(/N=N\c3ccc(Nc4ccccc4)c4c(S(=O)(=O)O)cccc34)cc(S(=O)(=O)O)cc2c1

nearest known ligand 0.91

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.91
THRB P10828 2/20 0.91
KMT2A Q03164 2/20 0.91
SNCA P37840 3/20 0.50
CHAT P28329 1/20 0.50
ENPP2 Q13822 1/20 0.49
CYP1A2 P05177 4/20 0.48
CYP2C9 P11712 3/20 0.48
MAPK1 P28482 2/20 0.48
DNASE1L3 Q13609 1/20 0.48
TTR P02766 1/20 0.47
FABP4 P15090 1/20 0.47
CCNA2 P20248 1/20 0.47
CDK2 P24941 1/20 0.47
MAPK14 Q16539 1/20 0.47
NR4A1 P22736 1/20 0.47
PRMT1 Q99873 1/20 0.45
NSD2 O96028 1/20 0.44
DUSP3 P51452 1/20 0.44
PTPN5 P54829 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Anazolene SCHEMBL1476742 0.95 MEN1 (1.00) MEN1THRBKMT2ASNCACHAT
Anazolene SCHEMBL29375317 0.95 MEN1 (1.00) MEN1THRBKMT2ASNCACHAT
Anazolene SCHEMBL29387597 0.95 MEN1 (1.00) MEN1THRBKMT2ASNCACHAT
Anazolene SCHEMBL11148088 0.95 MEN1 (1.00) MEN1THRBKMT2ASNCACHAT
Anazolene SCHEMBL26460213 0.95 MEN1 (1.00) MEN1THRBKMT2ASNCACHAT
Anazolene SCHEMBL23595 0.94 MEN1 (0.98) MEN1THRBKMT2ASNCACHAT
Anazolene SCHEMBL23594 0.83 KMT2A (0.76) MEN1THRBKMT2ASNCACHAT
Anazolene SCHEMBL29374551 0.83 KMT2A (0.76) MEN1THRBKMT2ASNCACHAT
Anazolene SCHEMBL1649427 0.83 KMT2A (0.76) MEN1THRBKMT2ASNCACHAT
SCHEMBL12177943 0.79 MEN1 (0.71) MEN1THRBKMT2ASNCACHAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230127304-A1 NEW INHIBITORS FOR THE KEAP1-NRF2 PROTEIN-PROTEIN INTERACTION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230127304-A1 NEW INHIBITORS FOR THE KEAP1-NRF2 PROTEIN-PROTEIN INTERACTION KEAP1, HMOX1, NFE2L2 MEN1 4181/4885THRB 3076/4885KMT2A 2474/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.