SCHEMBL2662872

SCHEMBL2662872

O=C(C#Cc1ccccc1)c1ccc2ccccc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.60
ALDH1A1 P00352 5/20 0.54
HSP90AA1 P07900 4/20 0.54
MAPT P10636 4/20 0.54
NPSR1 Q6W5P4 3/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
OPRK1 P41145 2/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
HTT P42858 2/20 0.54
MITF O75030 1/20 0.54
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
PTPN1 P18031 1/20 0.50
PIN1 Q13526 1/20 0.50
ASIC3 Q9UHC3 1/20 0.47
S1PR2 O95136 1/20 0.47
KDM4E B2RXH2 2/20 0.46
HPGD P15428 2/20 0.46
NPC1 O15118 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30114938 1.00 VCP (0.60) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL10625119 0.83 VCP (0.81) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL9124703 0.82 HSP90AA1 (0.69) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL978641 0.79 VCP (0.75) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL3798644 0.79 VCP (0.59) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL28738494 0.78 VCP (0.58) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL8650544 0.78 VCP (0.58) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL28972916 0.78 VCP (0.67) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL21318361 0.77 ASIC3 (0.45) VCPALDH1A1HSP90AA1MAPTNPSR1
SCHEMBL28509442 0.77 ASIC3 (0.45) VCPALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115677739-A Preparation method of O, O-boron difluoride complex 华南理工大学 2023-02-03 CN disclosed
US-7799818-B2 Pyrazole derivatives, compositions containing such compounds and methods of use MERCK SHARP & DOHME CORP. (US) 2010-09-21 US disclosed
US-7598285-B2 Pyrazole derivatives, compositions containing such compounds and methods of use MERCK & CO., INC (US) 2009-10-06 US disclosed
US-20090176854-A1 N-[4-((1S)-1-{3-(3,5-Dichlorophenyl)-5-[6-(trifluoromethoxy)-2-naphthyl]-1H-pyrazol-1-yl}ethyl)benzoyl]- beta -alanine; type 2 diabetes, hyperglycemia, or insulin resistance MERCK SHARP & DOHME LLC 2009-07-09 US disclosed
US-20050272794-A1 Pyrazole derivatives, compositions containing such compounds and methods of use MERCK SHARP & DOHME LLC 2005-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050272794-A1 Pyrazole derivatives, compositions containing such compounds and methods of use PC, GOT2, PNLIP VCP 3233/4885ALDH1A1 1729/4885HSP90AA1 3577/4885
US-20090176854-A1 N-[4-((1S)-1-{3-(3,5-Dichlorophenyl)-5-[6-(trifluoromethoxy)-2-naphthyl]-1H-pyrazol-1-yl}ethyl)benzoyl]- beta -alanine; type 2 diabetes, hyperglycemia, or insulin resistance GOT2, GOT1, IAPP VCP 3287/4885ALDH1A1 800/4885HSP90AA1 2130/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.