SCHEMBL26664258

SCHEMBL26664258

Cc1cn2nc(C(=O)O)cc(C)c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.45
APOBEC3A P31941 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
KDM4E B2RXH2 8/20 0.39
SMPD3 Q9NY59 1/20 0.38
ALDH1A1 P00352 7/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
HIF1A Q16665 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 2/20 0.33
GAA P10253 2/20 0.33
KDM6B O15054 1/20 0.33
TET3 O43151 1/20 0.33
KDM4A O75164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31497245 0.87 SMPD3 (0.40) RXFP1KDM4ESMPD3ALDH1A1HPGD
SCHEMBL31082622 0.85 LMNA (0.41) RXFP1KDM4ESMPD3ALDH1A1HPGD
SCHEMBL31600992 0.83 KMT2A (0.41) KDM4ESMPD3ALDH1A1HPGDHSD17B10
SCHEMBL26664189 0.81 RXFP1 (0.35) RXFP1KDM4ESMPD3ALDH1A1HPGD
SCHEMBL26978235 0.80 ASPH (0.41) APOBEC3AAPOBEC3GKDM4EALDH1A1HSD17B10
SCHEMBL3755198 0.77 APOBEC3A (0.49) RXFP1APOBEC3AAPOBEC3GKDM4EALDH1A1
SCHEMBL22445908 0.77 APOBEC3A (0.41) RXFP1APOBEC3AAPOBEC3GKDM4EALDH1A1
SCHEMBL3970342 0.76 KDM4E (0.52) KDM4ESMPD3ALDH1A1HPGDHSD17B10
SCHEMBL28524393 0.75 APOBEC3A (0.41) RXFP1APOBEC3AAPOBEC3GKDM4EALDH1A1
SCHEMBL25151525 0.75 KDM4E (0.45) KDM4ESMPD3ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250353841-A1 HETEROCYCLIC COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE HUFF SARAH ELIZABETH (US) 2025-11-20 US disclosed
WO-2025111409-A1 HETEROCYCLIC COMPOUNDS OF FORMULA (I) FOR USE IN THE TREATMENT OF SPINAL MUSCULAR ATROPHY VIA MODULATION OF SMN2 SPLICING BIOGEN MA INC. (US) 2025-05-30 WO disclosed
WO-2025111547-A1 2,3-DIHYDROPYROLLOPYRIDINE CARBOXAMIDE COMPOUNDS AND METHODS OF USE THEREOF RGENTA THERAPEUTICS, INC. (US) 2025-05-30 WO disclosed
EP-4308572-B1 NEW THIENOPYRIMIDINONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2025-04-23 EP disclosed
CN-119866329-A Heterocyclic compounds for the treatment of huntington's disease 渤健马萨诸塞州股份有限公司 2025-04-22 CN disclosed
EP-4526292-A1 HETEROCYCLIC COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE Biogen MA Inc. (US) 2025-03-26 EP disclosed
WO-2024182788-A1 COMPOUNDS AND METHODS FOR MODULATING SPLICING REMIX THERAPEUTICS INC. (US) 2024-09-06 WO disclosed
US-20240182493-A1 PROCESS HOFFMANN-LA ROCHE INC. (US) 2024-06-06 US disclosed
EP-4308572-A1 NEW THIENOPYRIMIDINONE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2024-01-24 EP disclosed
EP-4308578-A2 PROCESS FOR PREPARING RISDIPLAM F. Hoffmann-La Roche AG (CH) 2024-01-24 EP disclosed
US-20240002407-A1 THIENOPYRIMIDINONE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2024-01-04 US disclosed
WO-2023225244-A1 HETEROCYCLIC COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE BIOGEN MA INC. (US) 2023-11-23 WO disclosed
WO-2023225244-A1 HETEROCYCLIC COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE BIOGEN MA INC. (US) 2023-11-23 WO disclosed
CN-117050096-A Preparation method of risperidone 杭州诺澳生物医药科技有限公司 2023-11-14 CN disclosed
CN-117015546-A Process for preparing Li Sipu blue 豪夫迈·罗氏有限公司 2023-11-07 CN disclosed
CN-116997555-A Novel thienopyrimidinone derivatives 豪夫迈·罗氏有限公司 2023-11-03 CN disclosed
WO-2022194800-A1 NEW THIENOPYRIMIDINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2022-09-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250353841-A1 HETEROCYCLIC COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE HTT, HYPK, ATXN2 RXFP1 4463/4885APOBEC3A 4200/4885APOBEC3G 4446/4885
US-20240002407-A1 THIENOPYRIMIDINONE DERIVATIVES XDH, P2RX4, TBXA2R RXFP1 309/4885APOBEC3A 4369/4885APOBEC3G 4363/4885
US-20240182493-A1 PROCESS CYP3A7, UGT2B7, UGT1A7 RXFP1 3836/4885APOBEC3A 1011/4885APOBEC3G 386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.