SCHEMBL26807679

SCHEMBL26807679

CC(C)c1c(C(F)(F)F)c2cc(CN3CCC(c4ccccc4)CC3)ccc2n(C)c1=O

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.45
DRD4 P21917 4/20 0.45
SIGMAR1 Q99720 2/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PARP1 P09874 3/20 0.43
TLR9 Q9NR96 1/20 0.41
TLR8 Q9NR97 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
GRM2 Q14416 4/20 0.40
MCHR1 Q99705 2/20 0.40
USP2 O75604 1/20 0.40
DRD3 P35462 1/20 0.40
CCR2 P41597 2/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26817280 0.88 MCHR1 (0.40) DRD4SIGMAR1GRM2MCHR1DRD3
SCHEMBL26817271 0.77 HRH3 (0.40) SIGMAR1
SCHEMBL26817286 0.75 HTR1A (0.37) DRD2SIGMAR1
SCHEMBL26817285 0.74 GRM2 (0.38) GRM2MCHR1USP2KCNH2
SCHEMBL26817278 0.73 HTR1A (0.36) SIGMAR1KCNH2
SCHEMBL22016170 0.72 KIF11 (0.42) MEN1KMT2ATLR9
SCHEMBL22017134 0.71 ATM (0.38) MEN1KMT2A
SCHEMBL26815145 0.68 AR (0.39) USP2
SCHEMBL4331832 0.66 LMNA (0.50) DRD2DRD4MEN1KMT2AGRM2
SCHEMBL1002852 0.65 MEN1 (0.81) DRD2DRD4SIGMAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023220741-A1 ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF DICE MOLECULES SV, INC. (US) 2023-11-16 WO disclosed