SCHEMBL26817285

SCHEMBL26817285

CC(C)c1c(C(F)(F)F)c2ccc(CN3CCC(F)(F)CC3)cc2n(C)c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.38
HRH3 Q9Y5N1 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
OPRL1 P41146 3/20 0.34
HSD11B1 P28845 1/20 0.34
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
PARG Q86W56 1/20 0.33
USP2 O75604 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DGKZ Q13574 2/20 0.33
OPRM1 P35372 1/20 0.32
KCNH2 Q12809 1/20 0.32
MCHR1 Q99705 1/20 0.32
HTR6 P50406 1/20 0.32
TACR1 P25103 1/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26817286 0.83 HTR1A (0.37) HRH3PARG
SCHEMBL26817278 0.80 HTR1A (0.36) PARGOPRM1KCNH2
SCHEMBL26817280 0.79 MCHR1 (0.40) GRM2HRH3KCNH2MCHR1HTR6
SCHEMBL26807679 0.74 DRD2 (0.45) GRM2USP2KCNH2MCHR1
SCHEMBL26817271 0.73 HRH3 (0.40) HRH3L3MBTL1
SCHEMBL26817066 0.72 ALDH1A1 (0.46) USP2
SCHEMBL22016170 0.71 KIF11 (0.42) L3MBTL1
SCHEMBL22017134 0.68 ATM (0.38)
SCHEMBL26815145 0.65 AR (0.39) USP2
SCHEMBL12160960 0.65 ALDH1A1 (0.54) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023220741-A1 ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF DICE MOLECULES SV, INC. (US) 2023-11-16 WO disclosed