SCHEMBL26817280

SCHEMBL26817280

CC(C)c1c(C(F)(F)F)c2cc(CN3CCC(F)CC3)ccc2n(C)c1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 10/20 0.40
KCNH2 Q12809 6/20 0.38
HRH3 Q9Y5N1 1/20 0.38
ACHE P22303 1/20 0.37
ENPP2 Q13822 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR6 P50406 1/20 0.36
DRD4 P21917 2/20 0.35
SIGMAR1 Q99720 2/20 0.35
DRD3 P35462 1/20 0.35
GRM2 Q14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26807679 0.88 DRD2 (0.45) MCHR1KCNH2DRD4SIGMAR1DRD3
SCHEMBL26817271 0.82 HRH3 (0.40) HRH3ACHESIGMAR1
SCHEMBL26817286 0.79 HTR1A (0.37) HRH3SIGMAR1
SCHEMBL26817285 0.79 GRM2 (0.38) MCHR1KCNH2HRH3HTR6GRM2
SCHEMBL26817278 0.78 HTR1A (0.36) KCNH2SIGMAR1
SCHEMBL22017134 0.75 ATM (0.38) ALDH1A1
SCHEMBL26815145 0.72 AR (0.39) ALDH1A1
SCHEMBL22016170 0.71 KIF11 (0.42) ALDH1A1
SCHEMBL22017359 0.67 KDM4E (0.36) ALDH1A1
SCHEMBL26817066 0.65 ALDH1A1 (0.46) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023220741-A1 ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF DICE MOLECULES SV, INC. (US) 2023-11-16 WO disclosed