SCHEMBL27375281

SCHEMBL27375281

CN1CCN(c2cccc3c2C(N)CCC3)CC1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.45
DRD2 P14416 3/20 0.43
DRD3 P35462 3/20 0.43
NCF1 P14598 1/20 0.41
DRD4 P21917 2/20 0.39
HTR1A P08908 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
CXCR4 P61073 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27546919 0.84 HTR2C (0.42) DRD2DRD3NCF1HTR1AHTR2A
SCHEMBL27546910 0.78 ADRA2C (0.37) ADRA2CDRD2DRD3NCF1DRD4
SCHEMBL27567085 0.76 ADRA2C (0.36) ADRA2CDRD2NCF1HTR2A
SCHEMBL16308828 0.76 ACHE (0.39) DRD2HTR1A
SCHEMBL2856023 0.76 ACHE (0.39) DRD2HTR1A
SCHEMBL27546915 0.74 DRD2 (0.41) ADRA2CDRD2DRD3NCF1DRD4
SCHEMBL7470810 0.73 CXCR4 (0.44) CXCR4
SCHEMBL7246237 0.73 NCF1 (0.36) ADRA2CDRD2DRD3NCF1DRD4
SCHEMBL7025288 0.72 DRD3 (0.47) ADRA2CDRD2DRD3CXCR4
SCHEMBL4788557 0.72 DRD3 (0.47) ADRA2CDRD2DRD3CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1073101-C Substituted 1,2,3, 4-tetrahydronaphthalene derivatives ASTRA AB (SE) 2001-10-17 CN disclosed
CN-1278727-A Monoamine oxidase inhibitors and h 5-ht1BCombinations of antagonists or partial agonists ASTRAZENECA AB (SE) 2001-01-03 CN disclosed
CN-1219170-A Substituted 1,2,3, 4-tetrahydronaphthalene derivatives ASTRA AB (SE) 1999-06-09 CN disclosed