SCHEMBL27477137

SCHEMBL27477137

CCCCc1cc(N)c(C(=O)OCc2ccccc2)c(=O)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.46
TSHR P16473 2/20 0.46
MAPK1 P28482 2/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP3A4 P08684 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
RAB9A P51151 4/20 0.45
NPC1 O15118 2/20 0.45
KMT2A Q03164 2/20 0.45
PARP1 P09874 1/20 0.44
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
MMP12 P39900 2/20 0.41
MMP1 P03956 1/20 0.41
PRKCZ Q05513 2/20 0.41
MAPT P10636 1/20 0.40
STAT1 P42224 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
POLB P06746 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27433280 0.81 RAB9A (0.50) TDP1MAPK1ALDH1A1RAB9ANPC1
SCHEMBL9530581 0.79 TDP1 (0.56) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL8884936 0.78 GPR84 (0.50) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL27492019 0.75 ALDH1A1 (0.41) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL949772 0.71 NPC1 (0.51) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL8885939 0.70 ALDH1A1 (0.51) TSHRALDH1A1L3MBTL1NPC1KMT2A
SCHEMBL7723904 0.70 ALDH1A1 (0.54) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL9339127 0.70 TNKS (0.45) L3MBTL1MAPTSMN1; SMN2LMNA
SCHEMBL7736627 0.69 ALDH1A1 (0.53) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL20656207 0.69 MMP2 (0.47) TDP1MAPK1ALDH1A1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1192035-C Inhibitors of interleukin-1'beta' converting enzyme VERTEX PHARMA (US) 2005-03-09 CN disclosed