SCHEMBL27486965

SCHEMBL27486965

COC(=O)c1ccc(C(=O)OC(C)(C)C)nc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.41
ALDH1A1 P00352 6/20 0.41
GAA P10253 5/20 0.41
GLA P06280 3/20 0.41
HSD17B10 Q99714 3/20 0.41
HPGD P15428 3/20 0.41
MAPT P10636 2/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
ATM Q13315 1/20 0.41
CFTR P13569 2/20 0.40
ATR Q13535 1/20 0.40
ABL1 P00519 1/20 0.40
TSHR P16473 2/20 0.37
LMNA P02545 1/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
CA5A P35218 1/20 0.36
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14956928 0.87 ALDH1A1 (0.47) KDM4EALDH1A1GAAGLAHSD17B10
SCHEMBL27473142 0.86 GABRA1 (0.40) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL14967079 0.81 ALDH1A1 (0.45) KDM4EALDH1A1GAAGLAHSD17B10
SCHEMBL13853239 0.79 CYP1A2 (0.54) KDM4EALDH1A1HSD17B10MAPTTSHR
SCHEMBL5264558 0.78 CYP1A2 (0.53) KDM4EALDH1A1GAAHSD17B10HPGD
SCHEMBL27907009 0.78 KDM4E (0.44) KDM4EALDH1A1GAAGLAHSD17B10
SCHEMBL27622981 0.77 KDM4E (0.47) KDM4EALDH1A1GAAGLAHSD17B10
SCHEMBL20306004 0.75 ALDH1A1 (0.49) KDM4EALDH1A1GAAGLAHSD17B10
SCHEMBL28251522 0.75 CA12 (0.35) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL27459666 0.74 ALDH1A1 (0.49) KDM4EALDH1A1HSD17B10HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117658893-A Method for carrying out cis-trans selective hydrogenation on 2, 5-substituted pyridine derivative by utilizing micro-packed bed 南京药石科技股份有限公司 2024-03-08 CN disclosed
CN-1210267-C 2-hydroxy-mutilin carbamate derivatives for antibacterial use SMITHKLINE BEECHAM PLC (GB) 2005-07-13 CN disclosed
CN-1427827-A 2-Hydroxy-mutilin carbamate derivatives for antibacterial use SMITHKLINE BEECHAM PLC (GB) 2003-07-02 CN disclosed