SCHEMBL276286

SCHEMBL276286

O=C(c1cc(Cl)c[nH]1)C(Cl)(Cl)Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.60
HPGD P15428 2/20 0.60
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.48
PKM P14618 1/20 0.48
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
DYRK1A Q13627 1/20 0.41
DAO P14920 2/20 0.41
GRN P28799 1/20 0.40
SORT1 Q99523 1/20 0.40
NOTUM Q6P988 1/20 0.38
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPC1 O15118 1/20 0.33
TPMT P51580 1/20 0.32
RAB9A P51151 1/20 0.32
F7 P08709 1/20 0.31
F3 P13726 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1518124 0.78 ALDH1A1 (0.53) ALDH1A1HPGDLMNAGAAPKM
SCHEMBL13505930 0.78 ALDH1A1 (0.51) ALDH1A1HPGDLMNAGAAPKM
SCHEMBL2513855 0.78 ALDH1A1 (0.51) ALDH1A1HPGDLMNAGAAPKM
SCHEMBL600362 0.76
SCHEMBL4091668 0.75 ALDH1A1 (0.49) ALDH1A1HPGDLMNAGAAPKM
SCHEMBL1504448 0.75 ALDH1A1 (0.61) ALDH1A1HPGDLMNAGAAPKM
SCHEMBL261286 0.75 ALDH1A1 (0.49) ALDH1A1HPGDLMNAGAAPKM
SCHEMBL2148876 0.74
SCHEMBL276048 0.74
SCHEMBL3013942 0.73 ALDH1A1 (0.47) ALDH1A1HPGDLMNAGAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114456099-A Preparation method of 4-chloropyrrole-2-carboxylic acid 八叶草健康产业研究院(厦门)有限公司 2022-05-10 CN claimed
EP-4655069-A1 PYRIDAZINES AS SARM1 INHIBITORS Disarm Therapeutics, Inc. (US) 2025-12-03 EP disclosed
US-20250171434-A1 SEC61 INHIBITORS AND USE THEREOF ENODIA THERAPEUTICS SAS (FR) 2025-05-29 US disclosed
EP-4486451-A1 SEC61 INHIBITORS AND USE THEREOF Kezar Life Sciences, Inc. (US) 2025-01-08 EP disclosed
EP-4426699-A1 ANTHELMINTIC PYRROLOPYRIDAZINE COMPOUNDS Boehringer Ingelheim Vetmedica GmbH (DE) 2024-09-11 EP disclosed
WO-2024158775-A1 PYRIDAZINES AS SARM1 INHIBITORS DISARM THERAPEUTICS, INC. (US) 2024-08-02 WO disclosed
US-20240254133-A1 ANTHELMINTIC PYRROLOPYRIDAZINE COMPOUNDS BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2024-08-01 US disclosed
CN-118339164-A Insect repellent pyrrolopyridazine compounds 勃林格殷格翰动物保健有限公司 2024-07-12 CN disclosed
US-11999742-B2 Substituted pyrrolo[1,2-b]pyridazines as anthelmintics BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2024-06-04 US disclosed
WO-2023073641-A9 ANTHELMINTIC PYRROLOPYRIDAZINE COMPOUNDS BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2024-02-29 WO disclosed
US-20090209523-A1 Pyrrolo[1,2-A] Pyrazin-1(2H)-One and Pyrrolo[1,2-D][1,2,4]Triazin-1(2H)-One Derivatives as Inhibitors of Poly(Adp-Ribose)Polymerase (Parp) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2009-08-20 US disclosed
US-20090209523-A1 Pyrrolo[1,2-A] Pyrazin-1(2H)-One and Pyrrolo[1,2-D][1,2,4]Triazin-1(2H)-One Derivatives as Inhibitors of Poly(Adp-Ribose)Polymerase (Parp) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2009-08-20 US disclosed
US-20090203737-A1 Pyrrole Derivatives as Positive Allosteric Modulators of Metabotropic Receptors ADDEX PHARMA SA (CH) 2009-08-13 US disclosed
EP-2032140-A1 PYRROLO[1,2-A]PYRAZIN-1(2H)-ONE AND PYRROLO[1,2-D][1,2,4]TRIAZIN-1(2H)-ONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE(PARP) Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2009-03-11 EP disclosed
EP-1957077-A2 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS Bayer HealthCare LLC (US) 2008-08-20 EP disclosed
EP-1912979-A2 PHENYL-3-{(3-(1H-PYRROL-2-YL)-[1,2,4]OXADIAZOL-5-YL]PIPERIDIN-1-YL}-METHANONE DERIVATIVES AND RELATED COMPOUNDS AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX Pharma S.A. (CH) 2008-04-23 EP disclosed
WO-2007138355-A1 PYRROLO[1,2-A]PYRAZIN-1(2H)-ONE AND PYRROLO[1,2-D][1,2,4]TRIAZIN-1(2H)-ONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE(PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-12-06 WO disclosed
WO-2007064883-A2 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER HEALTHCARE LLC. (US) 2007-06-07 WO disclosed
WO-2007064883-A2 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER HEALTHCARE LLC. (US) 2007-06-07 WO disclosed
WO-2006123257-A2 PHENYL-3-{(3-(1H-PYRROL-2-YL)-[1, 2 , 4]0XADIAZ0L-5-YL]PIPERIDIN-1-YL}-METHANONE DERIVATIVES AND RELATED COMPOUNDS AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMA SA (CH) 2006-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250171434-A1 SEC61 INHIBITORS AND USE THEREOF SEC61B, SEC61A1, SEC61G ALDH1A1 4635/4885HPGD 1600/4885LMNA 2999/4885
US-20240254133-A1 ANTHELMINTIC PYRROLOPYRIDAZINE COMPOUNDS IL5, EPX, MPO ALDH1A1 1069/4885HPGD 578/4885LMNA 4215/4885
US-11999742-B2 Substituted pyrrolo[1,2-b]pyridazines as anthelmintics IL5, PLPBP, PNPO ALDH1A1 741/4885HPGD 501/4885LMNA 3481/4885
US-20090203737-A1 Pyrrole Derivatives as Positive Allosteric Modulators of Metabotropic Receptors GRM5, GRIK5, GRM2 ALDH1A1 4261/4885HPGD 2812/4885LMNA 4701/4885
US-20090209523-A1 Pyrrolo[1,2-A] Pyrazin-1(2H)-One and Pyrrolo[1,2-D][1,2,4]Triazin-1(2H)-One Derivatives as Inhibitors of Poly(Adp-Ribose)Polymerase (Parp) PARP1, PARP2, PARP11 ALDH1A1 139/4885HPGD 957/4885LMNA 1512/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.