SCHEMBL27656

SCHEMBL27656

CON(C)C(=O)c1cccnn1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.46
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
SNCA P37840 1/20 0.40
AHR P35869 1/20 0.38
FAAH O00519 1/20 0.38
CES1 P23141 1/20 0.37
TRPM8 Q7Z2W7 2/20 0.37
MLYCD O95822 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
TBXA2R P21731 1/20 0.35
CYP1A2 P05177 1/20 0.35
CLK1 P49759 1/20 0.34
DYRK1A Q13627 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
CTNNB1 P35222 1/20 0.33
WNT3A P56704 1/20 0.33
GAA P10253 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374828 0.82 P2RX7 (0.52) P2RX7KMT2AMEN1SNCAAHR
SCHEMBL6602091 0.78 P2RX7 (0.56) P2RX7KMT2AMEN1AHRFAAH
SCHEMBL8374791 0.78 KDM4E (0.45) KMT2AMEN1TRPM8MLYCDCYP1A2
SCHEMBL306106 0.77 ALDH1A1 (0.53) KMT2AMEN1CES1GAA
SCHEMBL27539765 0.77 P2RX7 (0.55) P2RX7KMT2AMEN1AHRFAAH
Hydrochloric Acid SCHEMBL29205819 0.77 P2RX7 (0.55) P2RX7KMT2AMEN1AHRFAAH
SCHEMBL30963925 0.74 P2RX7 (0.51) P2RX7FAAHCES1CTDSP1CYP1A2
SCHEMBL24724207 0.74 MLYCD (0.37) KMT2AMEN1FAAHTRPM8MLYCD
SCHEMBL30003812 0.74 MLYCD (0.37) KMT2AMEN1FAAHTRPM8MLYCD
SCHEMBL5026814 0.74 P2RX7 (0.55) P2RX7KMT2AMEN1SNCAAHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120040441-A Compositions and methods for treating cancer A2A制药有限公司 2025-05-27 CN disclosed
CN-119522217-A Compositions and methods for treating cancer A2A制药有限公司 2025-02-25 CN disclosed
EP-3938364-B1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES ALTERITY THERAPEUTICS LTD (AU) 2023-08-23 EP disclosed
EP-3938364-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES Alterity Therapeutics Limited (AU) 2022-01-19 EP disclosed
CN-113811533-A Compounds and methods for treating diseases 艾特里提治疗有限公司 2021-12-17 CN disclosed
US-10941143-B2 Imidazo [1,5-a]pyridine compounds and their use Alterity Therapeutics Limited (AU) 2021-03-09 US disclosed
US-10941143-B2 Imidazo [1,5-a]pyridine compounds and their use Alterity Therapeutics Limited (AU) 2021-03-09 US disclosed
WO-2020186291-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES Alterity Therapeutics Limited (AU) 2020-09-24 WO disclosed
US-20200291021-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES Alterity Therapeutics Limited (AU) 2020-09-17 US disclosed
US-20200291021-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES Alterity Therapeutics Limited (AU) 2020-09-17 US disclosed
US-8633212-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-01-21 US disclosed
US-8633212-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-01-21 US disclosed
US-8633212-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-01-21 US disclosed
EP-2406240-A2 INHIBITORS OF BETA-SECRETASE Vitae Pharmaceuticals, Inc. (US) 2012-01-18 EP disclosed
US-20110245224-A1 FUSED, SPIROCYCLIC HETEROAROMATIC COMPOUNDS FOR THE TREATMENT OF BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2011-10-06 US disclosed
US-20110071126-A1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. 2011-03-24 US disclosed
US-20110071126-A1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. 2011-03-24 US disclosed
US-20110071126-A1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. 2011-03-24 US disclosed
WO-2010105179-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-09-16 WO disclosed
WO-2010105179-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-09-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10941143-B2 Imidazo [1,5-a]pyridine compounds and their use SNCA, PARK7, HTT P2RX7 3381/4885KMT2A 654/4885MEN1 2116/4885
US-20110245224-A1 FUSED, SPIROCYCLIC HETEROAROMATIC COMPOUNDS FOR THE TREATMENT OF BACTERIAL INFECTIONS SDHB, SDHA, RORC P2RX7 2685/4885KMT2A 3960/4885MEN1 1594/4885
US-20200291021-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES SNCA, HTT, PARK7 P2RX7 4460/4885KMT2A 555/4885MEN1 1136/4885
US-20110071126-A1 INHIBITORS OF BETA-SECRETASE BACE1, BACE2, PSEN1 P2RX7 3251/4885KMT2A 3063/4885MEN1 905/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.