SCHEMBL2769756

SCHEMBL2769756

COC(CNCc1cc(Cl)cc2ccccc12)OC

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
SMPD1 P17405 1/20 0.36
DNM1 Q05193 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
MAPK1 P28482 1/20 0.35
MC5R P33032 1/20 0.35
PTGS2 P35354 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MITF O75030 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27650320 0.79 BCHE (0.43) MEN1KMT2ASMN1; SMN2MAPK1MC5R
SCHEMBL4153142 0.76 IFNAR1 (0.45) PTGS2
SCHEMBL2771330 0.74 CASR (0.37) SMN1; SMN2CYP2D6
SCHEMBL13430504 0.72 KMT2A (0.49) MEN1KMT2ASMPD1DNM1MAPK1
SCHEMBL31227163 0.71 HTT (0.44) CYP1A2CYP2D6ALDH1A1
SCHEMBL2769396 0.71 POLB (0.38) MEN1KMT2ASMN1; SMN2DNM1CYP1A2
SCHEMBL5200340 0.70 TACR1 (0.34) MEN1KMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL28948705 0.70 PTGS2 (0.42) CYP1A2CYP2D6CYP2C19PTGS2ALDH1A1
SCHEMBL13576841 0.70 ACLY (0.47) MEN1KMT2ASMN1; SMN2CYP1A2CYP2C19
SCHEMBL19643755 0.70 HTT (0.43) MEN1KMT2ASMN1; SMN2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1753739-B1 IMIDAZOL-2-ONE COMPOUNDS USEFUL IN THE TREATMENT OF VARIOUS DISORDERS GLAXO GROUP LTD (GB) 2010-04-28 EP disclosed
US-7534893-B2 Imidazol-2-one compounds useful in the treatment of various disorders GLAXO GROUP LIMITED (GB) 2009-05-19 US disclosed
US-20070249679-A1 Imidazol-2-One Compounds Useful in the Treatment of Various Disorders GLAXO GROUP LIMITED (GB) 2007-10-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070249679-A1 Imidazol-2-One Compounds Useful in the Treatment of Various Disorders SLC6A4, SLC18A2, SLC18A1 MEN1 1835/4885KMT2A 2977/4885SMN1; SMN2 1787/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.