SCHEMBL27697694

SCHEMBL27697694

CC(C)(C)C(=O)ON1CCN(c2ccccc2Br)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
LMNA P02545 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
ALDH1A1 P00352 4/20 0.40
RBP4 P02753 4/20 0.40
MAPT P10636 3/20 0.40
HTT P42858 2/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
POLB P06746 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GLA P06280 2/20 0.37
KDM4E B2RXH2 1/20 0.37
DRD2 P14416 1/20 0.37
USP2 O75604 1/20 0.37
UCHL1 P09936 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28746134 0.79 GOT1 (0.33) MEN1KMT2ALMNAALDH1A1MAPT
SCHEMBL30062550 0.78 GPR119 (0.52) MEN1KMT2ALMNASMN1; SMN2ALDH1A1
SCHEMBL1928396 0.78 GPR119 (0.52) MEN1KMT2ALMNASMN1; SMN2ALDH1A1
SCHEMBL28762854 0.78 ADRA2C (0.39) MEN1KMT2ALMNASMN1; SMN2ALDH1A1
SCHEMBL28840342 0.75 POLB (0.42) MEN1KMT2ALMNASMN1; SMN2ALDH1A1
SCHEMBL30937462 0.72 ALDH1A1 (0.59) MEN1KMT2ALMNASMN1; SMN2ALDH1A1
SCHEMBL18600520 0.72 ALDH1A1 (0.59) MEN1KMT2ALMNASMN1; SMN2ALDH1A1
SCHEMBL28794456 0.71 MEN1 (0.39) MEN1KMT2ALMNASMN1; SMN2ALDH1A1
SCHEMBL25389057 0.71 NCF1 (0.55) MEN1KMT2AALDH1A1HTTHTR1A
SCHEMBL28866522 0.70 KDM4E (0.33) MEN1KMT2ALMNASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109912514-A (2- heteroaryl aminocarbonyl phenyl) azepine ring derivatives and application thereof 广东东阳光药业有限公司 2019-06-21 CN disclosed
CN-106458943-B Synthesis of vortioxetine via (2, 4-dimethylphenyl) (2-iodophenyl) sulfane intermediate 斯洛文尼亚莱柯制药股份有限公司 2019-05-03 CN disclosed
CN-106279071-B Phenylpiperazine derivatives and its application method and purposes 广东东阳光药业有限公司 2019-01-04 CN disclosed
CN-106458943-A Synthesis of vortioxetine via (2, 4-dimethylphenyl) (2-iodophenyl) sulfane intermediate 斯洛文尼亚莱柯制药股份有限公司 2017-02-22 CN disclosed
CN-106279071-A Phenylpiperazine derivatives and using method thereof and purposes 广东东阳光药业有限公司 2017-01-04 CN disclosed
CN-106103419-A Method for synthesizing vortioxetine through (2- (piperazine-1-yl) phenyl) aniline intermediate 斯洛文尼亚莱柯制药股份有限公司 2016-11-09 CN disclosed
CN-105939995-A Synthesis of vortioxetine via (2-(piperazine-1 -yl)phenvl)lithium intermediates 斯洛文尼亚莱柯制药股份有限公司 2016-09-14 CN disclosed
CN-105348204-A 1-heterocyclyl-2-(heteroarylthio) benzene derivative and use method and application RUYUAN YAO AUTONOMOUS COUNTY DAZHONG MEDICINE TRADING CO LTD 2016-02-24 CN disclosed
CN-105339361-A Novel process for the synthesis of 1- (2- ((2, 4-dimethylphenyl) thio) phenyl) piperazine LEK PHARMACEUTICALS 2016-02-17 CN disclosed
CN-105283442-A New process for the synthesis of 1-(2-((2,4-dimethylphenyl)thio)phenyl)piperazine LEK PHARMACEUTICALS 2016-01-27 CN disclosed
CN-104829558-A Preparation method for diaryl thioether amine compound JIANGSU HANSOH PHARMACEUTICAL 2015-08-12 CN disclosed
CN-101830867-A Preparation method of 2- (3,3,5, 5-tetramethylcyclohexyl) aniline EISAI R&D MAN CO LTD 2010-09-15 CN disclosed
CN-101146760-A Intermediate for producing [ 2- (3,3,5, 5-tetramethylcyclohexyl) phenyl ] piperazine compound EISAI R&D MAN CO LTD (JP) 2008-03-19 CN disclosed