SCHEMBL2776253

SCHEMBL2776253

CC(C)[C@H](NC(=O)O)C(=O)N1CCC(Oc2ncc(C(F)(F)F)cn2)CC1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 7/20 0.45
CCR1 P32246 6/20 0.41
HRH3 Q9Y5N1 2/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
EPHX2 P34913 1/20 0.40
KCNH2 Q12809 1/20 0.39
HMOX1 P09601 1/20 0.39
ENPP2 Q13822 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2778165 0.88 CCR1 (0.48) CCR1KCNH2HMOX1
SCHEMBL2774358 0.88 LIPE (0.59) LIPEHRH3EPHX2ENPP2
SCHEMBL2777053 0.86 CCR1 (0.48) CCR1KCNH2
SCHEMBL2776334 0.86 HMOX1 (0.53) CCR1KCNH2HMOX1
SCHEMBL2776929 0.84 LMNA (0.48) CCR1KCNH2HMOX1
SCHEMBL2779821 0.84 CCR1 (0.47) CCR1EPHX2KCNH2HMOX1
SCHEMBL2777291 0.84 EPHX2 (0.53) LIPECCR1EPHX2
SCHEMBL2773592 0.83 P2RX3 (0.46) LIPE
SCHEMBL2776114 0.82 ACACB (0.46) CCR1CYP3A4KCNH2HMOX1
SCHEMBL2774470 0.82 ACACB (0.44) CCR1CYP2C9EPHX2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258697-A1 HYDROXYQUINOXALINECARBOXAMIDE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2010-12-08 EP disclosed