SCHEMBL278328

SCHEMBL278328

COc1ccc(Oc2cccc(C(C)(C)C)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.55
SMN1; SMN2 Q16637 5/20 0.53
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
ALDH1A1 P00352 4/20 0.46
HTT P42858 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MAPT P10636 4/20 0.44
NPC1 O15118 2/20 0.44
MAPK1 P28482 2/20 0.44
RAB9A P51151 2/20 0.44
HPGD P15428 1/20 0.44
MTNR1B P49286 3/20 0.44
MTNR1A P48039 2/20 0.44
RAF1 P04049 1/20 0.43
POLB P06746 1/20 0.43
MEN1 O00255 1/20 0.42
MITF O75030 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13009187 0.91 SMN1; SMN2 (0.55) LTA4HSMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL13474891 0.89 MAPT (0.57) SMN1; SMN2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL18118971 0.88 CYP3A4 (0.59) SMN1; SMN2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL5671239 0.86 CYP2C9 (0.54) LTA4HSMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL146154 0.86 ACHE (0.52) SMN1; SMN2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL15576545 0.86 CYP3A4 (0.57) SMN1; SMN2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL13790956 0.85 SMN1; SMN2 (0.62) LTA4HSMN1; SMN2ALDH1A1HTTMAPT
SCHEMBL12293087 0.85 HTT (0.50) SMN1; SMN2CYP3A4CYP2C9CYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL29893927 0.84 ACHE (0.50) SMN1; SMN2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL1284070 0.84 ALDH1A1 (0.67) SMN1; SMN2CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8716491-B2 Benzimidazolium dyes and their use as fluorescent chemosensors NEW YORK UNIVERSITY (US) 2014-05-06 US disclosed
US-8133898-B2 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-13 US disclosed
US-8133898-B2 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-13 US disclosed
US-20110301192-A1 Inhibitors of Cyclin Kinase Inhibitor p21 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-12-08 US disclosed
US-20110224231-A1 Novel Lactams as Beta Secretase Inhibitors PFIZER INC. (US) 2011-09-15 US disclosed
US-7947712-B2 Antiarthritic agents; asthma; chronic obstructive pulminary diosrders; atherosclerosis; vision defects; hepatitis; central nervous system disorders; cardiovascular disorders; wound healing agents; restenosis; cirrhosis; multiple sclerosis; glomerulonephritis; graft versus host disease; antidiabetic agent WYETH LLC (US) 2011-05-24 US disclosed
US-20100137310-A1 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-03 US disclosed
US-20080269213-A1 8-Hydroxyquinoline compounds and methods thereof WYETH (US) 2008-10-30 US disclosed
US-20080160521-A1 BENZIMIDAZOLIUM DYES AND THEIR USE AS FLUORESCENT CHEMOSENSORS NEW YORK UNIVERSITY (US) 2008-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137310-A1 RENIN INHIBITORS REN, ACE, PRSS3 LTA4H 752/4885SMN1; SMN2 4780/4885CYP3A4 49/4885
US-20080269213-A1 8-Hydroxyquinoline compounds and methods thereof MMP8, MMP26, MMP9 LTA4H 288/4885SMN1; SMN2 598/4885CYP3A4 1436/4885
US-20080160521-A1 BENZIMIDAZOLIUM DYES AND THEIR USE AS FLUORESCENT CHEMOSENSORS IK, C9, CBR3 LTA4H 521/4885SMN1; SMN2 3488/4885CYP3A4 840/4885
US-20110301192-A1 Inhibitors of Cyclin Kinase Inhibitor p21 CDKN1A, CCNI, CDK2 LTA4H 3233/4885SMN1; SMN2 4021/4885CYP3A4 3206/4885
US-20110224231-A1 Novel Lactams as Beta Secretase Inhibitors BACE1, BACE2, APH1B LTA4H 657/4885SMN1; SMN2 361/4885CYP3A4 1254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.