SCHEMBL2787166

SCHEMBL2787166

C=CCc1cnc2[nH]c(-c3cccnc3N)c(-c3ccccc3)c2n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.34
CDK2 P24941 2/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
MAP4K4 O95819 1/20 0.32
CCNT1 O60563 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK9 P50750 1/20 0.32
CCNB2 O95067 2/20 0.32
CCNB1 P14635 2/20 0.32
GSK3A P49840 2/20 0.32
GSK3B P49841 2/20 0.32
CCNB3 Q8WWL7 2/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
AKT1 P31749 1/20 0.30
AKT2 P31751 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2787037 0.78 CDK5 (0.41) CDK1CDK2MAP4K4CDK9CCNB2
SCHEMBL2787754 0.69 CCNB2 (0.39) CDK1CCNB2CCNB1GSK3AGSK3B
SCHEMBL2216872 0.65 CDK1 (0.42) CDK1CDK2MKNK1MKNK2MAP4K4
SCHEMBL2786751 0.63 CCNB2 (0.49) CDK1CCNB2CCNB1GSK3AGSK3B
SCHEMBL1148699 0.61 MAP4K4 (0.66) CDK1CDK2MKNK1MKNK2MAP4K4
SCHEMBL1779054 0.61 CCNB2 (0.48) CDK1CCNB2CCNB1GSK3AGSK3B
SCHEMBL5312790 0.61 BACE1 (0.42)
SCHEMBL11212892 0.60 ADRB2 (0.39)
SCHEMBL27727264 0.60 MAPK1 (0.38) CDC7
SCHEMBL253273 0.59 LMNA (0.55) PDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046215-A2 DIAZA-INDOLE DERIVATIVES AND THEIR USE AS FUNGICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-04-29 WO disclosed