SCHEMBL27903763

SCHEMBL27903763

O=C(NNc1nncs1)Oc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.49
POLB P06746 4/20 0.45
KDM4E B2RXH2 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NR3C1 P04150 1/20 0.43
TSHR P16473 1/20 0.43
MIF P14174 2/20 0.42
KMT2A Q03164 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
LMNA P02545 1/20 0.40
MEN1 O00255 1/20 0.40
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2160439 0.85 TAAR1 (0.59) TAAR1POLBKDM4ECYP1A2CYP3A4
SCHEMBL27966122 0.76 TAAR1 (0.49) TAAR1POLBKDM4ECYP1A2CYP3A4
SCHEMBL9553582 0.72 GAA (0.58) KDM4ECYP1A2CYP3A4TSHRKMT2A
SCHEMBL27785586 0.72 GOT1 (0.40) POLBKDM4ECYP1A2MIFKMT2A
SCHEMBL27692836 0.71 GAA (0.68) KDM4ECYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL27851689 0.71 RAB9A (0.50) POLBKDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL28109363 0.69 LMNA (0.49) TAAR1POLBKDM4ECYP3A4TSHR
SCHEMBL27763680 0.69 ALDH1A1 (0.42) KDM4ECYP1A2KMT2AHTTSMN1; SMN2
SCHEMBL28849976 0.68 BCAT2 (0.46) KDM4ECYP1A2KMT2AHTTSMN1; SMN2
SCHEMBL27716616 0.68 GAA (0.55) KDM4EKMT2AHTTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103415520-A Pyrrolo six-membered heteroaromatic ring derivative, preparation method thereof and application thereof in medicines JIANGSU HENGRUI MEDICINE CO 2013-11-27 CN disclosed
CN-102822177-A Pyrrolo [ 2, 3 - d] pyrimidine urea compounds as jak inhibitors PFIZER 2012-12-12 CN disclosed