SCHEMBL28008356

SCHEMBL28008356

Cc1cc(-c2[c]ccc(C(F)(F)F)c2)ccn1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 9/20 0.43
PSEN2 P49810 9/20 0.43
APH1B Q8WW43 9/20 0.43
NCSTN Q92542 9/20 0.43
APH1A Q96BI3 9/20 0.43
PSENEN Q9NZ42 9/20 0.43
CYP2D6 P10635 5/20 0.42
GRM2 Q14416 2/20 0.38
CYP3A4 P08684 1/20 0.38
S1PR1 P21453 1/20 0.38
TDO2 P48775 1/20 0.38
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
DYRK1A Q13627 1/20 0.37
SORT1 Q99523 1/20 0.37
PDK2 Q15119 1/20 0.36
NR2E1 Q9Y466 2/20 0.36
RORA P35398 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7024108 0.80 DYRK1A (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8078513 0.79 KIF11 (0.52) S1PR1NOS3NOS2
SCHEMBL17392954 0.78 CTSS (0.39) GRM2NOS3NOS2
SCHEMBL2296580 0.76 RAPGEF4 (0.35) CYP3A4
SCHEMBL16055751 0.76 NPBWR1 (0.41) CYP3A4
SCHEMBL5897973 0.75 PTPN5 (0.41)
SCHEMBL28007985 0.75 SORT1 (0.38) NOS3NOS2DYRK1ASORT1
SCHEMBL29497390 0.74 NOS3 (0.57) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1312951 0.74 NOS3 (0.57) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14258707 0.74 PSEN1 (0.59) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104394869-A Substituted bicyclic aza-heterocycles and analogues as sirtuin modulators GLAXOSMITHKLINE LLC 2015-03-04 CN disclosed