SCHEMBL28028277

SCHEMBL28028277

O=C(Nc1ccc2[nH]c(C(=O)NNc3ccccc3)cc2c1)c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.63
MAOB P27338 1/20 0.63
EGFR P00533 6/20 0.62
PIK3CA P42336 6/20 0.62
TP53 P04637 1/20 0.60
POLB P06746 1/20 0.60
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
LMNA P02545 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
NHERF1 O14745 2/20 0.59
PIN1 Q13526 1/20 0.56
MAPT P10636 1/20 0.55
JAK2 O60674 1/20 0.53
PTGS2 P35354 1/20 0.51
PYGL P06737 1/20 0.50
KCNK3 O14649 1/20 0.50
KCNK9 Q9NPC2 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28229577 0.88 TP53 (0.56) MAOAMAOBEGFRPIK3CATP53
SCHEMBL10466165 0.85 MAOA (0.71) MAOAMAOBEGFRPIK3CATP53
SCHEMBL28028254 0.85 MAOA (0.66) MAOAMAOBEGFRPIK3CATP53
SCHEMBL7533561 0.79 NPC1 (0.74) MAOAMAOBEGFRPIK3CATP53
SCHEMBL8205048 0.79 NHERF1 (0.64) MAOAMAOBEGFRPIK3CATP53
SCHEMBL27690981 0.79 MAOA (0.72) MAOAMAOBEGFRPIK3CATP53
SCHEMBL2760086 0.79 NPC1 (0.73) EGFRPIK3CATP53POLBNPC1
SCHEMBL27325791 0.78 MAOA (0.60) MAOAMAOBEGFRPIK3CATP53
SCHEMBL29429724 0.78 MAOB (1.00) MAOAMAOBTP53POLBNPC1
SCHEMBL24601450 0.77 MMP13 (0.72) MAOAMAOBEGFRPIK3CATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104860866-B 5- (substitution carbon acylamino) -1H- indoles -2- carbohydrazide derivatives and its preparation method and application 厦门大学 2018-07-17 CN disclosed
CN-104860866-A 5-(substituted carbonylamino)-1H-indole-2-carbohydrazide derivatives as well as preparation method and application thereof UNIV XIAMEN 2015-08-26 CN disclosed