SCHEMBL28032753

SCHEMBL28032753

CC(=O)NNc1cccc(CN)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.55
TSHR P16473 2/20 0.55
ALOX5 P09917 1/20 0.55
LOXL2 Q9Y4K0 1/20 0.49
ENPP2 Q13822 1/20 0.47
HTR6 P50406 1/20 0.45
GAA P10253 1/20 0.45
CFD P00746 1/20 0.44
NOS1 P29475 4/20 0.44
NOS2 P35228 4/20 0.44
ALDH1A1 P00352 4/20 0.42
NOS3 P29474 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NFKB1 P19838 1/20 0.42
CYP1A2 P05177 2/20 0.42
NPSR1 Q6W5P4 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
AOC3 Q16853 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2545099 0.83 ALDH1A1 (0.61) TSHRLOXL2CFDALDH1A1SMN1; SMN2
SCHEMBL28032259 0.82 CYP3A4 (0.57) CYP3A4TSHRALOX5LOXL2GAA
Hydrochloric Acid SCHEMBL1127877 0.81 ALDH1A1 (0.59) TSHRLOXL2CFDALDH1A1CYP1A2
SCHEMBL20027769 0.77 HTR6 (0.47) CYP3A4LOXL2ENPP2HTR6CFD
SCHEMBL5708790 0.77 ALDH1A1 (0.69) CYP3A4TSHRALOX5GAAALDH1A1
SCHEMBL19119342 0.77 LOXL2 (0.49) CYP3A4TSHRLOXL2ENPP2HTR6
SCHEMBL28141068 0.76 MTNR1A (0.61) CYP3A4TSHRLOXL2HTR6CFD
SCHEMBL8648511 0.75 GAA (0.76) CYP3A4TSHRALOX5GAAALDH1A1
SCHEMBL3003205 0.74 CFD (0.59) TSHRLOXL2ENPP2HTR6GAA
SCHEMBL2557430 0.74 CFD (0.55) TSHRLOXL2ENPP2HTR6GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104945403-A Tetrahydrobenzo [ e ] [1,2,4] triaza compounds and preparation method thereof UNIV DALIAN TECH 2015-09-30 CN disclosed