SCHEMBL28032764

SCHEMBL28032764

O=Cc1cc(Br)ccc1-c1ccc[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.44
CYP2A6 P11509 3/20 0.42
PIM3 Q86V86 2/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
PIM1 P11309 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP2D6 P10635 2/20 0.33
CYP1B1 Q16678 2/20 0.33
AURKA O14965 1/20 0.33
KDR P35968 1/20 0.33
S100A4 P26447 1/20 0.33
PTPRC P08575 1/20 0.33
PTPN1 P18031 1/20 0.33
CDK2 P24941 1/20 0.33
CYP1A2 P05177 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
IDO1 P14902 1/20 0.32
CHEK1 O14757 1/20 0.32
WEE1 P30291 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL203395 0.78 ERN1 (0.61) ERN1CYP2A6PIM3PTGDR2PIM1
SCHEMBL30239797 0.77 MEN1 (0.46) CYP2A6ALDH1A1AURKAKDRCDK2
SCHEMBL5961899 0.77 MEN1 (0.46) CYP2A6ALDH1A1AURKAKDRCDK2
SCHEMBL28032258 0.75 ERN1 (0.50) ERN1ALDH1A1CYP2D6S100A4PTPRC
SCHEMBL31167504 0.74 GPR35 (0.44) CYP2A6ALDH1A1AURKAKDRS100A4
SCHEMBL1985834 0.72 ERN1 (0.50) ERN1CYP2A6PTGDR2ALDH1A1S100A4
SCHEMBL27814203 0.71 S100A4 (0.47) ERN1ALDH1A1S100A4
SCHEMBL16050049 0.70 ERN1 (0.48) ERN1CYP2A6PTGDR2ALDH1A1S100A4
SCHEMBL30214858 0.70 IMPDH2 (0.49) PIM3PIM1AURKACDK2IDO1
SCHEMBL405754 0.68 ALDH1A1 (0.47) ERN1CYP2A6PIM3PTGDR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104945403-A Tetrahydrobenzo [ e ] [1,2,4] triaza compounds and preparation method thereof UNIV DALIAN TECH 2015-09-30 CN disclosed