SCHEMBL28047000

SCHEMBL28047000

COc1ccc(Cn2nnc(C(=O)O)c2Oc2cccc(OC)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 9/20 0.55
HCAR3 P49019 1/20 0.49
MAPT P10636 2/20 0.48
POLB P06746 2/20 0.48
ALOX15 P16050 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ALDH1A1 P00352 2/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
AKR1C2 P52895 1/20 0.45
HSD17B10 Q99714 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21296984 0.91 AKR1C3 (0.49) AKR1C3HCAR3MAPTPOLBALOX15
SCHEMBL22815682 0.91 AKR1C3 (0.47) AKR1C3HCAR3MAPTPOLBALOX15
SCHEMBL22816536 0.90 AKR1C3 (0.47) AKR1C3HCAR3MAPTPOLBALOX15
SCHEMBL21296988 0.90 NPC1 (0.48) AKR1C3HCAR3MAPTPOLBALOX15
SCHEMBL29891535 0.89 AKR1C3 (0.47) AKR1C3HCAR3MAPTPOLBALOX15
SCHEMBL22815906 0.88 ALOX15 (0.47) AKR1C3MAPTPOLBALOX15L3MBTL1
SCHEMBL28047047 0.87 CYP19A1 (0.50) AKR1C3MAPTPOLBALOX15L3MBTL1
SCHEMBL21296968 0.87 AKR1C3 (0.46) AKR1C3HCAR3MAPTPOLBALOX15
SCHEMBL21296920 0.86 NPBWR1 (0.51) AKR1C3MAPTPOLBALOX15L3MBTL1
SCHEMBL22815761 0.86 CCR2 (0.50) AKR1C3MAPTPOLBALOX15L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164112-A Amide compound and preparation method, pharmaceutical composition and application thereof SHANGHAI INST MATERIA MEDICA 2015-12-16 CN disclosed