SCHEMBL28053239

SCHEMBL28053239

CCOc1ncc(S(N)(=O)=O)cc1-c1cncc(Cl)c1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.38
CA1 P00915 5/20 0.36
CA2 P00918 5/20 0.36
CA9 Q16790 5/20 0.36
CA12 O43570 3/20 0.36
CA14 Q9ULX7 2/20 0.36
RORC P51449 1/20 0.35
BRD4 O60885 1/20 0.35
KMT2A Q03164 1/20 0.35
PTGS1 P23219 5/20 0.35
PTGS2 P35354 5/20 0.35
CA7 P43166 2/20 0.35
ALDH1A1 P00352 3/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
CCNA1 P78396 2/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
AURKA O14965 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28826183 0.88 APLNR (0.40) APLNRCA1CA2CA9CA12
SCHEMBL28053242 0.81 APLNR (0.43) APLNRCA1CA2CA9PTGS1
SCHEMBL28826194 0.81 SOS1 (0.39) APLNRCA1CA2CA9CA12
SCHEMBL28053258 0.74 PKM (0.46) APLNRCA1CA2CA9CA12
SCHEMBL28053374 0.74 LRRK2 (0.44) APLNRCA1CA2CA9CA12
SCHEMBL28053310 0.73 SCN10A (0.44) APLNRCA1CA2CA9CA12
SCHEMBL28053322 0.72 APLNR (0.51) APLNRCA1CA2CA9CA12
SCHEMBL28053327 0.71 APLNR (0.45) APLNRCA1CA2CA9CA12
SCHEMBL16235621 0.70 S100A9 (0.49) RORCKMT2AALDH1A1NPSR1LMNA
SCHEMBL28053234 0.68 NPSR1 (0.41) CA1CA2CA9CA12KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN claimed
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed