SCHEMBL28053258

SCHEMBL28053258

NS(=O)(=O)c1ccc(-c2cncc(Cl)c2O)c(-c2cncc(Cl)c2O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
TDP2 O95551 1/20 0.43
NSD2 O96028 1/20 0.43
HK1 P19367 1/20 0.43
PAX8 Q06710 1/20 0.43
CA1 P00915 9/20 0.43
CA2 P00918 9/20 0.43
CA9 Q16790 9/20 0.43
CA12 O43570 6/20 0.42
CA7 P43166 2/20 0.42
CA14 Q9ULX7 2/20 0.42
APLNR P35414 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA5B Q9Y2D0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053374 0.87 LRRK2 (0.44) TDP2NSD2HK1PAX8CA1
SCHEMBL28053244 0.81 RORC (0.44) CA1CA2CA9PTGS1PTGS2
SCHEMBL28053242 0.79 APLNR (0.43) CA1CA2CA9APLNRPTGS1
SCHEMBL28053327 0.79 APLNR (0.45) POLBCA1CA2CA9CA12
SCHEMBL28053322 0.78 APLNR (0.51) POLBALDH1A1CA1CA2CA9
SCHEMBL28826183 0.76 APLNR (0.40) CA1CA2CA9CA12CA7
SCHEMBL28053310 0.76 SCN10A (0.44) ALDH1A1GAAMAPTCA1CA2
SCHEMBL28826194 0.74 SOS1 (0.39) MAPTCA1CA2CA9CA12
SCHEMBL28053239 0.74 APLNR (0.38) POLBALDH1A1CA1CA2CA9
SCHEMBL28053341 0.73 PKM (0.49) PKMPOLBALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed